SCHEMBL2359893

SCHEMBL2359893

C=C[CH]N1C(=O)C=CC1=O

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 4/20 0.35
GSK3A P49840 1/20 0.35
GSK3B P49841 1/20 0.35
FAAH O00519 2/20 0.32
GMNN O75496 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
THPO P40225 1/20 0.31
BLM P54132 1/20 0.31
PMP22 Q01453 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1664700 0.77
SCHEMBL28572221 0.69 MGLL (0.42) MGLLGSK3AGSK3BFAAHGMNN
SCHEMBL1389139 0.69
SCHEMBL5457531 0.65 ALDH1A1 (0.46) GSK3BALDH1A1MAPTNPSR1
SCHEMBL28379307 0.65
SCHEMBL9777831 0.65
SCHEMBL22916701 0.64 GMNN (0.30) MGLLGMNNALDH1A1LMNAMAPT
SCHEMBL15577150 0.63 MGLL (0.38) MGLLGSK3AGSK3BFAAHGMNN
SCHEMBL4978013 0.62 GAA (0.31) MGLLGSK3AGSK3B
Butadiene SCHEMBL11308511 0.62 MGLL (0.42) MGLLGSK3AGSK3BFAAHGMNN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024067295-A1 MODIFIED RED BLOOD CELL AND USE THEREOF FOR DELIVERING MEDICAMENT 西湖生物医药科技(杭州)有限公司 2024-04-04 WO claimed
EP-1590373-B1 CONJUGATES OBTAINED BY REDUCTIVE AMINATION OF SEROTYPE 5 PNEUMOCOCCUS CAPSULAR POLYSACCHARIDE SANOFI PASTEUR (FR) 2011-08-17 EP claimed
EP-1590373-A1 CONJUGATES OBTAINED BY REDUCTIVE AMINATION OF SEROTYPE 5 PNEUMOCOCCUS CAPSULAR POLYSACCHARIDE Sanofi Pasteur (FR) 2005-11-02 EP claimed
WO-2004067574-A1 CONJUGATES OBTAINED BY REDUCTIVE AMINATION OF SEROTYPE 5 PNEUMOCOCCUS CAPSULAR POLYSACCHARIDE SANOFI PASTEUR (FR) 2004-08-12 WO claimed
WO-2024067295-A1 MODIFIED RED BLOOD CELL AND USE THEREOF FOR DELIVERING MEDICAMENT 西湖生物医药科技(杭州)有限公司 2024-04-04 WO disclosed
EP-1590373-B1 CONJUGATES OBTAINED BY REDUCTIVE AMINATION OF SEROTYPE 5 PNEUMOCOCCUS CAPSULAR POLYSACCHARIDE SANOFI PASTEUR (FR) 2011-08-17 EP disclosed
EP-1590373-A1 CONJUGATES OBTAINED BY REDUCTIVE AMINATION OF SEROTYPE 5 PNEUMOCOCCUS CAPSULAR POLYSACCHARIDE Sanofi Pasteur (FR) 2005-11-02 EP disclosed
WO-2004067574-A1 CONJUGATES OBTAINED BY REDUCTIVE AMINATION OF SEROTYPE 5 PNEUMOCOCCUS CAPSULAR POLYSACCHARIDE SANOFI PASTEUR (FR) 2004-08-12 WO disclosed
US-6361777-B1 COVALENTLY COUPLING POLYSACCHARIDE TO BIOPOLYMER HAVING HYDROXYL, AMINO AND/OR MERCAPTO GROUPS BY ACTIVATING POLYSACCHARIDE WITH CYANOGEN BROMIDE, THIOLATING WITH AMINOTHIOL LINKER, REACTING WITH BIOPOLYMER DE STAAT DER NEDERLANDEN,VERTEGENWOORDIGD DOOR DE MINISTER VAN WELZIJN, VOLKSGEZONDHEID EN CULTUUR (NL) 2002-03-26 US disclosed
EP-1163273-A1 METHOD FOR THE REDUCTIVE ANIMATION OF POLYSACCHARIDES Aventis Pasteur (FR) 2001-12-19 EP disclosed
EP-0848011-B1 Method of coupling polysaccharides to proteins NEDERLANDEN STAAT (NL) 2001-03-21 EP disclosed
WO-2000055210-A1 METHOD FOR THE REDUCTIVE AMINATION OF POLYSACCHARIDES AVENTIS PASTEUR (FR) 2000-09-21 WO disclosed
EP-1035137-A1 Method for the reductive amination of polysaccharides PASTEUR MERIEUX SERUMS ET VACCINS (FR) 2000-09-13 EP disclosed
WO-1998027107-A1 METHOD OF COUPLING POLYSACCHARIDES TO PROTEINS DE STAAT DER NEDERLANDEN, VERTEGENWOORDIGD DOOR DE MINISTER VAN WELZIJN, VOLKSGEZONDHEID EN CULTUUR (NL) 1998-06-25 WO disclosed
EP-0848011-A1 Method of coupling polysaccharides to proteins DE STAAT DER NEDERLANDEN VERTEGENWOORDIGD DOOR DE MINISTER VAN WELZIJN, VOLKSGEZONDHEID EN CULTUUR (NL) 1998-06-17 EP disclosed
US-4855468-A Titanocenes and a radiation-polymerizable composition containing these titanocenes CIBA-GEIGY CORPORATION (US) 1989-08-08 US disclosed
US-4713401-A PHOTOINITIATORS ORTHO-CF2Z GROUP CIBA SPECIALTY CHEMICALS CORPORATION 1987-12-15 US disclosed