SCHEMBL23600216

SCHEMBL23600216

C=C(/C=C(\C)C(N)=O)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.45
CYP2C19 P33261 2/20 0.45
MAPT P10636 2/20 0.45
TSHR P16473 2/20 0.45
TDP1 Q9NUW8 2/20 0.45
POLB P06746 1/20 0.45
CYP3A4 P08684 1/20 0.45
RECQL P46063 1/20 0.45
BLM P54132 1/20 0.45
PMP22 Q01453 1/20 0.45
HSD17B10 Q99714 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
CES2 O00748 2/20 0.42
CES1 P23141 2/20 0.42
GAA P10253 1/20 0.41
AKT1 P31749 1/20 0.41
ALDH1A1 P00352 3/20 0.41
LMNA P02545 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3386465 0.84 AKR1C3 (0.50) PARP1MAPTTSHRTDP1MEN1
SCHEMBL21182922 0.83 MEN1 (0.39) PARP1CYP2C19MAPTTSHRTDP1
SCHEMBL3794069 0.82 NFE2L2 (0.55) PARP1CYP2C19MAPTTSHRTDP1
SCHEMBL3794074 0.82 NFE2L2 (0.55) PARP1CYP2C19MAPTTSHRTDP1
SCHEMBL23268276 0.82 KMT2A (0.39) PARP1CYP2C19MAPTTSHRTDP1
SCHEMBL6258204 0.77 MEN1 (0.42) MAPTTSHRTDP1MEN1KMT2A
SCHEMBL24254437 0.77 MEN1 (0.42) MAPTTSHRTDP1CYP3A4MEN1
SCHEMBL12907944 0.75 BLM (0.41) PARP1CYP2C19MAPTTSHRTDP1
SCHEMBL10479693 0.75 DEGS1 (0.43) MAPTMEN1KMT2ACES2CES1
SCHEMBL19141920 0.75 DEGS1 (0.43) MAPTMEN1KMT2ACES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021130255-A1 DIHYDRO-CYCLOPENTA-ISOQUINOLINE DERIVATIVES UCB Biopharma SRL (BE) 2021-07-01 WO disclosed