SCHEMBL23602

SCHEMBL23602

Cc1nc(C)c(C(=O)Nc2ccccc2)s1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 1.00
RECQL P46063 1/20 1.00
NPC1 O15118 5/20 0.75
MAPT P10636 5/20 0.75
SMN1; SMN2 Q16637 6/20 0.74
TP53 P04637 1/20 0.74
ALDH1A1 P00352 7/20 0.64
HTT P42858 5/20 0.64
CYP1A2 P05177 1/20 0.64
CYP3A4 P08684 1/20 0.64
CYP2C9 P11712 1/20 0.64
LMNA P02545 3/20 0.61
KDM4E B2RXH2 3/20 0.60
GAA P10253 1/20 0.59
MEN1 O00255 5/20 0.59
KMT2A Q03164 5/20 0.59
NPSR1 Q6W5P4 2/20 0.59
HPGD P15428 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11651472 0.85 RAB9A (1.00) RAB9ARECQLNPC1MAPTSMN1; SMN2
SCHEMBL5135408 0.84 RAB9A (0.73) RAB9ARECQLNPC1MAPTSMN1; SMN2
SCHEMBL11714015 0.84 RAB9A (0.73) RAB9ARECQLNPC1MAPTSMN1; SMN2
SCHEMBL774205 0.84 MAPT (0.81) RAB9ARECQLNPC1MAPTSMN1; SMN2
SCHEMBL42334 0.84 RAB9A (0.97) RAB9ARECQLNPC1MAPTSMN1; SMN2
SCHEMBL27971154 0.84 F10 (0.73) RAB9ARECQLNPC1MAPTSMN1; SMN2
SCHEMBL8302044 0.83 RAB9A (0.71) RAB9ARECQLNPC1MAPTSMN1; SMN2
SCHEMBL27971290 0.83 RAB9A (0.70) RAB9ARECQLNPC1MAPTSMN1; SMN2
SCHEMBL2519126 0.83 RAB9A (0.70) RAB9ARECQLNPC1MAPTSMN1; SMN2
SCHEMBL15836431 0.82 RAB9A (0.69) RAB9ARECQLNPC1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 7582 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3060043-B1 PESTICIDAL COMPOSITIONS AND RELATED METHODS CORTEVA AGRISCIENCE LLC (US) 2025-11-26 EP claimed
EP-3578542-B1 COMPOSITIONS HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-11-12 EP claimed
EP-4646109-A2 NATURAL LIPID PARTICLE FORMULATIONS FOR AGRICULTURAL APPLICATIONS Invaio Sciences, Inc. (US) 2025-11-12 EP claimed
EP-3578543-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-08-20 EP claimed
US-12391729-B2 Fusion proteins, recombinant bacteria, and methods for using recombinant bacteria SPOGEN BIOTECH INC. (US) 2025-08-19 US claimed
EP-3578541-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY, AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-05-28 EP claimed
US-12163142-B2 Methods for manufacturing plant messenger packs FLAGSHIP PIONEERING INNOVATIONS VI, LLC (US) 2024-12-10 US claimed
WO-2024168193-A2 NATURAL LIPID PARTICLE FORMULATIONS FOR AGRICULTURAL APPLICATIONS INVAIO SCIENCES, INC. (US) 2024-08-15 WO claimed
US-20240199709-A1 FUSION PROTEINS, RECOMBINANT BACTERIA, AND METHODS FOR USING RECOMBINANT BACTERIA SPOGEN BIOTECH INC (US) 2024-06-20 US claimed
US-20240188569-A1 NEW YEAST STRAIN AND ITS USES FOR THE CONTROL OF PHYTOPATHOGENS AGROVENTURES LLC (US) 2024-06-13 US claimed
CN-1812715-A Active substance combinations with nematicidal, insecticidal and fungicidal properties based on trifluorobutenyl compounds BAYER CROPSCIENCE AG (DE) 2006-08-02 CN claimed
EP-1453817-B1 THIAZOLE DERIVATIVES WITH FUNGICIDAL ACTIVITY ISAGRO RICERCA SRL (IT) 2006-04-26 EP claimed
EP-1622453-A1 ACTIVE SUBSTANCE COMBINATIONS THAT HAVE NEMATICIDAL, INSECTICIDAL, AND FUNGICIDAL PROPERTIES AND ARE BASED ON TRIFLUOROBUTENYL COMPOUNDS Bayer CropScience AG (DE) 2006-02-08 EP claimed
US-20050065197-A1 Thiazole derivatives with fungicidal activity ISAGRO RICERCA S.R.L. (IT) 2005-03-24 US claimed
WO-2004095929-A1 ACTIVE SUBSTANCE COMBINATIONS THAT HAVE NEMATICIDAL, INSECTICIDAL, AND FUNGICIDAL PROPERTIES AND ARE BASED ON TRIFLUOROBUTENYL COMPOUNDS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2004-11-11 WO claimed
EP-1453817-A1 THIAZOLE DERIVATIVES WITH FUNGICIDAL ACTIVITY Isagro Ricerca S.r.l. (IT) 2004-09-08 EP claimed
WO-2003050096-A1 THIAZOLE DERIVATIVES WITH FUNGICIDAL ACTIVITY ISAGRO RICERCA S.R.L. (IT) 2003-06-19 WO claimed
WO-2001056358-A2 ENHANCED PROPERTIED PESTICIDES ROHM AND HAAS COMPANY (US) 2001-08-09 WO claimed
US-5730996-A Intercalates and expoliates formed with organic pesticide compounds and compositions containing the same AMCOL INTERNATIONAL CORPORATION (US) 1998-03-24 US claimed
US-5468747-A Fungicidal compositions and methods of use employing pyrimidine derivatives ZENECA LIMITED (GB) 1995-11-21 US claimed