SCHEMBL23608697

SCHEMBL23608697

CC(C)(C)OC(=O)Nc1cc(F)nc(C(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.39
CYP17A1 P05093 3/20 0.38
TOP2A P11388 1/20 0.36
TOP2B Q02880 1/20 0.36
EGLN2 Q96KS0 3/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA9 Q16790 1/20 0.36
PSMB8 P28062 1/20 0.36
NAMPT P43490 1/20 0.36
MAP4K4 O95819 1/20 0.36
APLNR P35414 1/20 0.35
AAK1 Q2M2I8 1/20 0.35
SMARCA2 P51531 1/20 0.35
LCK P06239 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25839112 0.84 CYP17A1 (0.38) SYKCYP17A1TOP2ATOP2BEGLN2
SCHEMBL30013712 0.84 CYP17A1 (0.38) SYKCYP17A1TOP2ATOP2BEGLN2
SCHEMBL29883076 0.79 SYK (0.39) SYKCYP17A1TOP2ATOP2BEGLN2
SCHEMBL23608484 0.79 SYK (0.39) SYKCYP17A1TOP2ATOP2BEGLN2
SCHEMBL18820155 0.78 SMARCA2 (0.59) SYKCYP17A1CA12CA1CA9
SCHEMBL31042935 0.78 CYP17A1 (0.40) SYKCYP17A1TOP2ATOP2BEGLN2
SCHEMBL23580147 0.77 SMARCA2 (0.37) SMARCA2
SCHEMBL30493119 0.77 BACE1 (0.35) SYKCYP17A1TOP2ATOP2BCA12
SCHEMBL31745657 0.77 BACE1 (0.35) SYKCYP17A1TOP2ATOP2BCA12
SCHEMBL25839110 0.77 BACE1 (0.35) SYKCYP17A1TOP2ATOP2BCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114945571-B Cyclic compounds and methods of use thereof 薛定谔公司 2025-02-25 CN disclosed
US-20240018157-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME SCHRÖDINGER, INC. 2024-01-18 US disclosed
US-20240018157-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME SCHRÖDINGER, INC. 2024-01-18 US disclosed
US-20240018157-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME SCHRÖDINGER, INC. 2024-01-18 US disclosed
EP-4081526-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME Schrödinger, Inc. (US) 2022-11-02 EP disclosed
CN-114945571-A Cyclic compounds and methods of use thereof 薛定谔公司 2022-08-26 CN disclosed
WO-2021134004-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME SCHRODINGER, INC. (US) 2021-07-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240018157-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME MALT1, FKBP1B, FKBP1A SYK 240/4885CYP17A1 353/4885TOP2A 1229/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.