SCHEMBL23622263

SCHEMBL23622263

CC(C)C(COc1ccc2[nH]ncc2c1)NC(=O)C(C)(F)F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
POLB P06746 1/20 0.43
NPC1 O15118 4/20 0.42
RAB9A P51151 3/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ROCK2 O75116 7/20 0.42
KCNH2 Q12809 1/20 0.40
ROCK1 Q13464 5/20 0.39
XDH P47989 1/20 0.39
MAPK1 P28482 1/20 0.38
MAOB P27338 1/20 0.37
CLK2 P49760 1/20 0.37
BLK P51451 1/20 0.37
CSNK2A1 P68400 1/20 0.37
STK3 Q13188 1/20 0.37
DYRK1A Q13627 1/20 0.37
AURKB Q96GD4 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
STK17A Q9UEE5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23622397 0.81 NR3C1 (0.44) MEN1KMT2ANPC1RAB9AL3MBTL1
SCHEMBL23622254 0.81 NPC1 (0.42) MEN1KMT2APOLBNPC1RAB9A
SCHEMBL21182244 0.79 NR3C1 (0.43) NPC1RAB9AROCK2ROCK1
SCHEMBL23622255 0.77 NR3C1 (0.43) MEN1KMT2ANPC1RAB9AL3MBTL1
SCHEMBL23622154 0.76 NR3C1 (0.55)
SCHEMBL17644001 0.76 NR3C1 (0.61)
SCHEMBL19459958 0.76 NR3C1 (0.61)
SCHEMBL23622136 0.76 NR3C1 (0.47) ROCK2
SCHEMBL23622250 0.75 NR3C1 (0.57)
SCHEMBL5407397 0.74 KCNH2 (0.49) MEN1KMT2ANPC1RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021136429-A1 BENZOPYRAZOLE COMPOUND 南京明德新药研发有限公司 2021-07-08 WO disclosed