SCHEMBL23628980

SCHEMBL23628980

COc1ccc(COc2c[nH]c(COc3cc(C(=O)O)cc4sc(NC(=O)c5cc(Br)c(Br)[nH]5)nc34)cc2=O)cc1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 2/20 0.51
CSNK2A2 P19784 3/20 0.43
CSNK2A1 P68400 3/20 0.43
SCD O00767 1/20 0.41
DUSP3 P51452 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23628961 0.96 TOP2A (0.46) TOP2ACSNK2A2CSNK2A1SCDDUSP3
SCHEMBL23628944 0.85 TOP2A (0.48) TOP2A
SCHEMBL23628962 0.85 SCD (0.48) TOP2ASCD
SCHEMBL23628936 0.83 TOP2A (0.46) TOP2ACSNK2A2CSNK2A1SCDDUSP3
SCHEMBL23629025 0.75 SCD (0.48) TOP2ASCD
SCHEMBL23943302 0.71
SCHEMBL23628899 0.70 TOP2A (0.90) TOP2A
SCHEMBL23628891 0.69
SCHEMBL23629049 0.68 MEN1 (0.42) SCD
SCHEMBL23628974 0.68 SCD (0.62) SCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12258342-B2 Class of DNA gyrase and/or topoisomerase IV inhibitors with activity against gram-positive and gram-negative bacteria UNIVERZA V LJUBLJANI (SI) 2025-03-25 US disclosed
US-20210323957-A1 NEW CLASS OF DNA GYRASE AND/OR TOPOISOMERASE IV INHIBITORS WITH ACTIVITY AGAINST GRAM-POSITIVE AND GRAM-NEGATIVE BACTERIA UNIVERZA V LJUBLJANI (SI) 2021-10-21 US disclosed
EP-3847172-A1 NEW CLASS OF DNA GYRASE AND/OR TOPOISOMERASE IV INHIBITORS WITH ACTIVITY AGAINST GRAM-POSITIVE AND GRAM-NEGATIVE BACTERIA Univerza v Ljubljani (SI) 2021-07-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210323957-A1 NEW CLASS OF DNA GYRASE AND/OR TOPOISOMERASE IV INHIBITORS WITH ACTIVITY AGAINST GRAM-POSITIVE AND GRAM-NEGATIVE BACTERIA TOP1, TOP2A, TOP2B TOP2A 2/4885CSNK2A2 814/4885CSNK2A1 630/4885
US-12258342-B2 Class of DNA gyrase and/or topoisomerase IV inhibitors with activity against gram-positive and gram-negative bacteria TOP1, TOP2A, TOP2B TOP2A 2/4885CSNK2A2 760/4885CSNK2A1 561/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.