SCHEMBL23629630

SCHEMBL23629630

C=CCc1cc(Br)cc2c(C(C)=O)nn(CC(=O)O)c12

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.36
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
MAPK1 P28482 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KRAS P01116 1/20 0.32
PTGDR2 Q9Y5Y4 2/20 0.30
PTGDR Q13258 1/20 0.30
CFD P00746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20488109 0.88 LMNA (0.41) LMNAKDM4EMEN1MAPK1KMT2A
SCHEMBL26679703 0.87 LMNA (0.40) LMNAKDM4EMEN1NPC1MAPK1
SCHEMBL23629634 0.87 LMNA (0.37) LMNAKDM4EMEN1NPC1MAPK1
SCHEMBL20488553 0.86 LMNA (0.33) LMNAKDM4EMEN1NPC1MAPK1
SCHEMBL26679590 0.85 LMNA (0.35) LMNAKDM4EMEN1NPC1MAPK1
SCHEMBL26679683 0.85 MTNR1A (0.31)
SCHEMBL20487966 0.85 LMNA (0.37) LMNAMEN1KMT2APTGDR2CFD
SCHEMBL20487312 0.84 LMNA (0.38) LMNAMEN1KMT2APTGDR2CFD
SCHEMBL26679658 0.84 LMNA (0.35) LMNAKDM4EMEN1NPC1MAPK1
SCHEMBL26679665 0.84 MAPT (0.36) LMNAKDM4EMEN1NPC1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3846803-A2 MACROCYCLIC COMPOUNDS FOR THE TREATMENT OF MEDICAL DISORDERS Achillion Pharmaceuticals, Inc. (US) 2021-07-14 EP disclosed