Sulfuric Acid

Sulfuric Acid

SCHEMBL2363547

COC(=O)c1ccc(CN)cc1.COC(=O)c1ccc(CN)cc1.O=S(=O)(O)O

nearest known ligand 0.86

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Sulfuric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 2/20 0.86
CA1 P00915 5/20 0.55
CA2 P00918 5/20 0.55
CA12 O43570 4/20 0.55
CA9 Q16790 4/20 0.55
CA14 Q9ULX7 4/20 0.55
MAPT P10636 2/20 0.55
CYP4A11 Q02928 2/20 0.53
STS P08842 1/20 0.53
HPGD P15428 1/20 0.51
CYP4F2 P78329 1/20 0.51
TDP1 Q9NUW8 1/20 0.50
HDAC3 O15379 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
NCOR2 Q9Y618 1/20 0.50
CA7 P43166 1/20 0.50
PTPRB P23467 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL184868 0.93 LOXL2 (1.00) LOXL2CA1CA2CA12CA9
Hydrochloric Acid SCHEMBL210547 0.91 LOXL2 (0.96) LOXL2CA1CA2CA12CA9
SCHEMBL6677665 0.87 LOXL2 (0.89) LOXL2CA1CA2CA12CA9
SCHEMBL28267713 0.84 LOXL2 (0.83) LOXL2CA1CA2CA12CA9
SCHEMBL12636516 0.84 LOXL2 (0.83) LOXL2CA1CA2CA12CA9
SCHEMBL7251467 0.84 LOXL2 (0.83) LOXL2CA1CA2CA12CA9
SCHEMBL21914682 0.84 LOXL2 (0.65) LOXL2CA1CA2CA12CA9
Sulfuric Acid SCHEMBL8295634 0.83 LOXL2 (0.59) LOXL2CA1CA2CA12CA9
SCHEMBL28117998 0.83 LOXL2 (0.80) LOXL2CA1CA2MAPTCYP4A11
Hydrochloric Acid SCHEMBL15239627 0.81 LOXL2 (0.77) LOXL2MAPTCYP4A11HPGDCYP4F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8008062-B2 Production of (R)- and (S)-4-(1-aminoethyl) benzoic acid methyl ester sulfate by lipase acylation of racemic 4-(1-aminoethyl) benzoic acid methyl ester and sulfuric acid precipitation BASF SE (DE) 2011-08-30 US claimed
CN-101321875-B Method for preparing -and (S) -methyl 4- (1-ammonioethyl) benzoate sulfate from racemic methyl 4- (1-aminoethyl) benzoate by lipase-catalyzed enantioselective acylation and subsequent precipitation with sulfuric acid BASF AG 2012-12-12 CN disclosed
EP-1969129-B1 PROCESS FOR THE PREPARATION OF (R)- AND (S)-4-(1-AMINOMETHYL) BENZOIC ACID METHYLESTER-SULPHATE FROM RACEMIC 4-(1-AMINOETHYL)BENZOIC ACID METHYLESTER BASF SE (DE) 2009-03-11 EP disclosed
US-20080305530-A1 Method for Producing (R)-and (S)-4-(1-Ammoniumethyl)Benzoic Acid Methylester-Sulphate from Racemic 4-(1-Aminoethyl)Benzoic Acid Methylester by Lipase Catalysed Enantoselective Acylation and Subsequent Precipitation with Sulphuric Acid BASF SE (DE) 2008-12-11 US disclosed
CN-101321875-A Method for preparing -and (S) -methyl 4- (1-ammonioethyl) benzoate sulfate from racemic methyl 4- (1-aminoethyl) benzoate by lipase-catalyzed enantioselective acylation and subsequent precipitation with sulfuric acid BASF AG (DE) 2008-12-10 CN disclosed
EP-1969129-A1 METHOD FOR PRODUCING (R) - AND (S)-4-(1-AMMONIUMETHYL)BENZOIC ACID METHYLESTER-SULPHATE FROM RACEMIC 4-(1-AMINOETHYL)BENZOIC ACID METHYLESTER BY LIPASE CATALYSED ENANTOSELECTIVE ACYLATION AND SUBSEQUENT PRECIPITATION WITH SULPHURIC ACID BASF SE (DE) 2008-09-17 EP disclosed
WO-2007077120-A1 METHOD FOR PRODUCING (R) - AND (S)-4-(1-AMMONIUMETHYL)BENZOIC ACID METHYLESTER-SULPHATE FROM RACEMIC 4-(1-AMINOETHYL)BENZOIC ACID METHYLESTER BY LIPASE CATALYSED ENANTOSELECTIVE ACYLATION AND SUBSEQUENT PRECIPITATION WITH SULPHURIC ACID BASF SE (DE) 2007-07-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080305530-A1 Method for Producing (R)-and (S)-4-(1-Ammoniumethyl)Benzoic Acid Methylester-Sulphate from Racemic 4-(1-Aminoethyl)Benzoic Acid Methylester by Lipase Catalysed Enantoselective Acylation and Subsequent Precipitation with Sulphuric Acid ARSA, APEH, STS LOXL2 1106/4885CA1 1615/4885CA2 1684/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.