SCHEMBL23636819

SCHEMBL23636819

CCS(=O)(=O)c1ccc(CNC(=O)c2ccc(N3CC[C@@H](Oc4ccc(C(F)(F)F)cc4)C3)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RORC P51449 13/20 0.52
ACACB O00763 5/20 0.47
MAPK14 Q16539 1/20 0.46
TP53 P04637 1/20 0.45
THRB P10828 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23632655 1.00 RORC (0.52) RORCACACBMAPK14TP53THRB
SCHEMBL23642189 0.93 RORC (0.53) RORCACACBMAPK14TP53THRB
SCHEMBL23636805 0.89 PRKAA2 (0.51) RORCACACB
SCHEMBL23636965 0.89 MEN1 (0.52) ACACBMAPK14
SCHEMBL23636728 0.89 DGAT2 (0.51) RORCACACB
SCHEMBL23636666 0.86 ACACB (0.47) ACACBMAPK14
SCHEMBL21619482 0.85 RORC (0.55) RORC
SCHEMBL21619519 0.85 RORC (0.55) RORC
SCHEMBL23632415 0.85 RORC (0.53) RORC
SCHEMBL23636932 0.85 RORC (0.49) RORCMAPK14TP53THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021139599-A1 RORγT INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF 东莞市东阳光新药研发有限公司 2021-07-15 WO disclosed