SCHEMBL23640290

SCHEMBL23640290

COc1ccc2c(ccc3oc(=O)cc(O)c32)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.59
EGFR P00533 1/20 0.53
KDM4E B2RXH2 7/20 0.53
ALDH1A1 P00352 6/20 0.53
HPGD P15428 5/20 0.53
HSD17B10 Q99714 3/20 0.53
CA12 O43570 2/20 0.53
CA1 P00915 2/20 0.53
CA3 P07451 2/20 0.53
CA4 P22748 2/20 0.53
CA5A P35218 2/20 0.53
CA7 P43166 2/20 0.53
CA9 Q16790 2/20 0.53
CA14 Q9ULX7 2/20 0.53
AKR1B1 P15121 1/20 0.53
CA6 P23280 1/20 0.53
CA2 P00918 1/20 0.51
CA5B Q9Y2D0 1/20 0.51
HNF4A P41235 1/20 0.48
NOD2 Q9HC29 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3911979 0.83 KDM4E (0.69) KDM4EALDH1A1HPGDHSD17B10CA12
SCHEMBL5341628 0.81 CYP2A6 (0.56) CYP2A6KDM4EALDH1A1HPGDHSD17B10
SCHEMBL3914588 0.80 KDM4E (0.69) CYP2A6KDM4EALDH1A1HPGDHSD17B10
SCHEMBL23640291 0.80 KDM4E (0.67) KDM4EALDH1A1HPGDHSD17B10CA12
SCHEMBL31026601 0.80 CYP2A6 (0.56) CYP2A6KDM4EALDH1A1HPGDHSD17B10
SCHEMBL23634920 0.80 DYRK1A (0.69) CYP2A6KDM4EALDH1A1HPGDHSD17B10
SCHEMBL29001886 0.79 CYP2A6 (0.76) CYP2A6KDM4EALDH1A1HPGDHSD17B10
SCHEMBL30450765 0.79 CYP2A6 (0.76) CYP2A6KDM4EALDH1A1HPGDHSD17B10
SCHEMBL23640303 0.78 ALDH1A1 (0.50) KDM4EALDH1A1HPGDHSD17B10CA12
SCHEMBL23640323 0.78 ALDH1A1 (0.50) KDM4EALDH1A1HPGDHSD17B10CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022262782-A1 GLUTARIMIDE-SUBSTITUTED ISOXAZOLE FUSED RING COMPOUND, AND APPLICATION THEREOF 南京明德新药研发有限公司 2022-12-22 WO disclosed
EP-3848367-A1 TRICYCLIC COMPOUNDS ACTING ON CRBN PROTEINS Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2021-07-14 EP disclosed