SCHEMBL23644684

SCHEMBL23644684

CC(C)(C)OC(=O)N(C1CCOCC1)n1cc(C(=O)O)c(=O)c2cc(Br)cnc21

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.35
OPRK1 P41145 3/20 0.34
BACE1 P56817 2/20 0.32
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20520865 0.89 PDE4B (0.47) PDE4BOPRK1
SCHEMBL25335713 0.81 LMNA (0.30)
SCHEMBL20520654 0.78 PDE4B (0.46) PDE4B
SCHEMBL29705143 0.78 PDE4B (0.46) PDE4B
SCHEMBL20520759 0.77 GSK3B (0.31) CNR2
SCHEMBL29705203 0.77 GSK3B (0.31) CNR2
SCHEMBL28735837 0.76 LMNA (0.33) BACE1
SCHEMBL27696252 0.73 HSD17B10 (0.36) OPRK1
SCHEMBL20240708 0.72 LMNA (0.34)
SCHEMBL23646765 0.70 LMNA (0.44) PDE4BOPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3601282-B1 NOVEL PYRIDO[2,3-B]INDOLE COMPOUNDS FOR THE TREATMENT AND PROPHYLAXIS OF BACTERIAL INFECTION HOFFMANN LA ROCHE (CH) 2021-07-21 EP disclosed