SCHEMBL29705143

SCHEMBL29705143

CCOC(=O)c1cn(N(C(=O)OC(C)(C)C)C2CCOCC2)c2ncc(B(O)O)cc2c1=O

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 10/20 0.46
HSD17B10 Q99714 3/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
USP2 O75604 1/20 0.36
TP53 P04637 1/20 0.36
MAPK1 P28482 1/20 0.36
RECQL P46063 1/20 0.36
PKM P14618 1/20 0.33
ADORA1 P30542 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
RAD52 P43351 1/20 0.32
UHRF1 Q96T88 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20520654 1.00 PDE4B (0.46) PDE4BHSD17B10KDM4EALDH1A1HPGD
SCHEMBL20520865 0.89 PDE4B (0.47) PDE4BHSD17B10KDM4EALDH1A1HPGD
SCHEMBL29705146 0.83 KDM4E (0.35) PDE4BHSD17B10KDM4EALDH1A1HPGD
SCHEMBL20521183 0.83 KDM4E (0.35) PDE4BHSD17B10KDM4EALDH1A1HPGD
SCHEMBL20521561 0.80 KDM4E (0.35) PDE4BHSD17B10KDM4EALDH1A1HPGD
SCHEMBL29705123 0.80 KDM4E (0.35) PDE4BHSD17B10KDM4EALDH1A1HPGD
SCHEMBL20521542 0.79 PDE4B (0.36) PDE4BPOLB
SCHEMBL23644684 0.78 PDE4B (0.35) PDE4B
SCHEMBL20521059 0.77 KDM4E (0.40) PDE4BHSD17B10KDM4EALDH1A1HPGD
SCHEMBL29705131 0.77 KDM4E (0.40) PDE4BHSD17B10KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110475777-B Novel pyrido [2,3-b ] indole compounds for the treatment and prevention of bacterial infections 豪夫迈·罗氏有限公司 2022-04-15 CN disclosed