SCHEMBL2364501

SCHEMBL2364501

CCCCCc1ccnc2ccccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 1/20 0.55
TLR8 Q9NR97 6/20 0.47
TLR7 Q9NYK1 2/20 0.46
S1PR2 O95136 1/20 0.45
LMNA P02545 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
CYP1A2 P05177 1/20 0.45
NCF1 P14598 1/20 0.44
KDM4E B2RXH2 1/20 0.44
USP2 O75604 1/20 0.44
ALDH1A1 P00352 1/20 0.44
GLA P06280 1/20 0.44
CYP3A4 P08684 1/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
CASP1 P29466 1/20 0.44
CASP7 P55210 1/20 0.44
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6115467 0.98 LOXL2 (0.53) LOXL2TLR8TLR7S1PR2LMNA
SCHEMBL6114494 0.98 LOXL2 (0.53) LOXL2TLR8TLR7S1PR2LMNA
SCHEMBL6114551 0.98 LOXL2 (0.53) LOXL2TLR8TLR7S1PR2LMNA
SCHEMBL6114968 0.98 LOXL2 (0.53) LOXL2TLR8TLR7S1PR2LMNA
SCHEMBL6114811 0.98 LOXL2 (0.53) LOXL2TLR8TLR7S1PR2LMNA
SCHEMBL6115139 0.98 LOXL2 (0.53) LOXL2TLR8TLR7S1PR2LMNA
SCHEMBL10585446 0.98 LOXL2 (0.53) LOXL2TLR8TLR7S1PR2LMNA
SCHEMBL6115140 0.98 LOXL2 (0.53) LOXL2TLR8TLR7S1PR2LMNA
SCHEMBL30665033 0.95 LOXL2 (0.56) LOXL2TLR8TLR7S1PR2LMNA
SCHEMBL2237676 0.95 LOXL2 (0.56) LOXL2TLR8TLR7S1PR2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 42 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113527198-A Method for preparing 4-arylquinoline from 2-aminodiaryl methanol 长沙资材科技有限公司 2021-10-22 CN claimed
CN-112047882-A New application of isoquinoline and quinoline derivatives in preparation of blood fat reducing drugs 天津科技大学 2020-12-08 CN claimed
CN-118324694-A Fluorescent compound for rapidly detecting explosive as well as preparation method and application thereof 湖南华南光电科技股份有限公司 2024-07-12 CN disclosed
CN-113527198-A Method for preparing 4-arylquinoline from 2-aminodiaryl methanol 长沙资材科技有限公司 2021-10-22 CN disclosed
CN-113527198-A Method for preparing 4-arylquinoline from 2-aminodiaryl methanol 长沙资材科技有限公司 2021-10-22 CN disclosed
CN-113527198-A Method for preparing 4-arylquinoline from 2-aminodiaryl methanol 长沙资材科技有限公司 2021-10-22 CN disclosed
US-10961266-B2 Chemoselective methylene hydroxylation in aromatic molecules THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2021-03-30 US disclosed
US-10961266-B2 Chemoselective methylene hydroxylation in aromatic molecules THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2021-03-30 US disclosed
CN-112047882-A New application of isoquinoline and quinoline derivatives in preparation of blood fat reducing drugs 天津科技大学 2020-12-08 CN disclosed
US-10654807-B2 Toll-like receptor 8 agonists THE UNIVERSITY OF KANSAS (US) 2020-05-19 US disclosed
US-20200087331-A1 CHEMOSELECTIVE METHYLENE HYDROXYLATION IN AROMATIC MOLECULES THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 2020-03-19 US disclosed
WO-2005033103-A1 QUINOLINE COMPOUNDS AND THEIR USES RIGEL PHARMACEUTICALS, INC. (US) 2005-04-14 WO disclosed
EP-0860433-B1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BREWERY (JP) 2002-07-03 EP disclosed
US-6388081-B1 4-substituted-quinoline derivatives and 4-substituted-quinoline combinatorial libraries LION BIOSCIENCE AG (DE) 2002-05-14 US disclosed
US-6262269-B1 4-Substituted-quinoline derivatives and 4-substituted-quinoline combinatorial libraries TREGA BIOSCIENCES, INC. 2001-07-17 US disclosed
US-6143764-A ETHER DERIVATIVES OF QUINOLINE, ANTITUMOR AGENTS KIRIN BEER KABUSHIKI KAISHA (JP) 2000-11-07 US disclosed
EP-0977989-A1 4-SUBSTITUTED-QUINOLINE DERIVATIVES AND 4-SUBSTITUTE-QUINOLINE COMBINATORIAL LIBRARIES TREGA BIOSCIENCES, INC. (US) 2000-02-09 EP disclosed
EP-0860433-A1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BEER KABUSHIKI KAISHA (JP) 1998-08-26 EP disclosed
WO-1998034115-A1 4-SUBSTITUTED-QUINOLINE DERIVATIVES AND 4-SUBSTITUTE-QUINOLINE COMBINATORIAL LIBRARIES TREGA BIOSCIENCES, INC. (US) 1998-08-06 WO disclosed
WO-1997048705-A1 POTASSIUM CHANNEL BLOCKERS UNIVERSITY COLLEGE LONDON (GB) 1997-12-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10654807-B2 Toll-like receptor 8 agonists TLR8, TLR7, TLR1 LOXL2 622/4885TLR8 1/4885TLR7 2/4885
US-10961266-B2 Chemoselective methylene hydroxylation in aromatic molecules PAH, DBH, AHR LOXL2 3162/4885TLR8 4000/4885TLR7 3874/4885
US-20200087331-A1 CHEMOSELECTIVE METHYLENE HYDROXYLATION IN AROMATIC MOLECULES PAH, DBH, AHR LOXL2 3162/4885TLR8 4000/4885TLR7 3874/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.