SCHEMBL23645561

SCHEMBL23645561

Nc1cc(-c2ccc(-c3ccccc3)cc2)cc(C(=O)O)c1N

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 2/20 0.56
KMT2A Q03164 4/20 0.55
KDM4E B2RXH2 3/20 0.55
GFER P55789 1/20 0.55
RXFP1 Q9HBX9 1/20 0.55
ACMSD Q8TDX5 3/20 0.55
MCL1 Q07820 3/20 0.55
HNF4A P41235 2/20 0.55
DHFR P00374 1/20 0.55
PTPN1 P18031 3/20 0.51
AKR1C2 P52895 3/20 0.50
AKR1C1 Q04828 3/20 0.50
AKR1C4 P17516 1/20 0.50
AKR1C3 P42330 1/20 0.50
PPM1B O75688 1/20 0.49
PTPN2 P17706 1/20 0.49
PTPN6 P29350 1/20 0.49
MEN1 O00255 3/20 0.48
USP2 O75604 2/20 0.48
MAPT P10636 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23645608 0.87 IKBKB (0.69) IKBKBKMT2AKDM4EGFERRXFP1
SCHEMBL23645723 0.82 ALDH1A1 (0.53) IKBKBKMT2AKDM4EMEN1MAPT
SCHEMBL12292220 0.81 PTPN1 (0.66) IKBKBKMT2AKDM4EACMSDMCL1
SCHEMBL30456877 0.81 PPM1B (0.71) IKBKBKMT2AKDM4EGFERRXFP1
SCHEMBL2575452 0.81 PPM1B (0.71) IKBKBKMT2AKDM4EGFERRXFP1
SCHEMBL2246915 0.81 KMT2A (0.84) IKBKBKMT2AKDM4EGFERRXFP1
SCHEMBL18176810 0.80 AKR1C2 (0.67) IKBKBKMT2AKDM4EGFERRXFP1
SCHEMBL27846422 0.80 KMT2A (0.59) IKBKBKMT2AKDM4EGFERRXFP1
SCHEMBL2426286 0.80 KDM4E (0.59) IKBKBKMT2AKDM4EGFERRXFP1
SCHEMBL23645564 0.78 PTPN1 (0.48) IKBKBKMT2AKDM4EGFERRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3915557-A1 METHODS OF USE FOR TRISUBSTITUTED BENZOTRIAZOLE DERIVATIVES AS DIHYDROOROTATE OXYGENASE INHIBITORS Aurigene Discovery Technologies Limited (IN) 2021-12-01 EP disclosed
EP-3615027-B1 METHODS OF USE FOR TRISUBSTITUTED BENZOTRIAZOLE DERIVATIVES AS DIHYDROOROTATE OXYGENASE INHIBITORS AURIGENE DISCOVERY TECH LTD (IN) 2021-07-14 EP disclosed