SCHEMBL2365254

SCHEMBL2365254

COC(=O)C=Cc1ccccc1NC(C)=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.56
CYP1A2 P05177 2/20 0.53
CYP2C9 P11712 2/20 0.53
CYP2C19 P33261 2/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
TSHR P16473 1/20 0.47
HPGD P15428 2/20 0.47
MAPT P10636 5/20 0.47
KDM4E B2RXH2 3/20 0.46
MEN1 O00255 1/20 0.46
TP53 P04637 1/20 0.46
ALOX15 P16050 1/20 0.46
KMT2A Q03164 1/20 0.46
HSD17B10 Q99714 1/20 0.46
NFE2L2 Q16236 1/20 0.44
SNCA P37840 2/20 0.44
TRPA1 O75762 1/20 0.44
TRPM8 Q7Z2W7 1/20 0.44
CA12 O43570 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL687505 1.00 ALDH1A1 (0.56) ALDH1A1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL1881446 1.00 ALDH1A1 (0.56) ALDH1A1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL27841557 0.87 SNCA (0.47) ALDH1A1CYP1A2CYP2C9CYP2C19HPGD
SCHEMBL29092108 0.86 ALDH1A1 (0.52) ALDH1A1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL11318756 0.86 CYP2C19 (0.49) ALDH1A1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL8740665 0.85 MAPT (0.55) ALDH1A1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL2779391 0.85 CYP2C19 (0.48) ALDH1A1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL7186932 0.83 CYP2C19 (0.55) ALDH1A1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL1881512 0.83 CYP2C19 (0.55) ALDH1A1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL2551111 0.83 CYP2C19 (0.55) ALDH1A1CYP1A2CYP2C9CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 67 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0954375-A4 NOVEL SUPPORTED CATALYSTS SETON HALL UNIVERSITY (US) 2000-06-21 EP claimed
US-6005148-A COMPRISING SUPPORT, ANCHORING AGENT SUCH AS HETEROPOLY ACID OR ANION, AND METAL COMPLEX USEFUL IN HYDROGENATION OF SUBSTITUTED UNSATURATED ACIDS AND ESTERS SETON HALL UNIVERSITY (US) 1999-12-21 US claimed
WO-1999064154-A1 POLY-OXYANIONS AS ANCHORING AGENTS FOR METAL COMPLEXES SETON HALL UNIVERSITY (US) 1999-12-16 WO claimed
EP-0954375-A1 NOVEL SUPPORTED CATALYSTS Seton Hall University (US) 1999-11-10 EP claimed
WO-1998028074-A1 NOVEL SUPPORTED CATALYSTS SETON HALL UNIVERSITY (US) 1998-07-02 WO claimed
CN-112824423-A Chiral ferrocenylphosphine-indolylaminophosphine ligand and preparation method and application thereof 中国科学院大连化学物理研究所 2021-05-21 CN disclosed
US-9884317-B2 Inorganic/polymeric hybrid catalytic materials with high activity in various solvents NIPPON KODOSHI CORPORATION (JP) 2018-02-06 US disclosed
US-9527067-B2 Inorganic/polymeric hybrid catalytic materials containing metal nano-particles therein NIPPON KODOSHI CORPORATION (JP) 2016-12-27 US disclosed
US-20150005154-A1 INORGANIC/POLYMERIC HYBRID CATALYTIC MATERIALS WITH HIGH ACTIVITY IN VARIOUS SOLVENTS NIPPON KODOSHI CORPORATION (JP) 2015-01-01 US disclosed
EP-2814607-A1 INORGANIC / POLYMERIC HYBRID CATALYTIC MATERIALS WITH HIGH ACTIVITY IN VARIOUS SOLVENTS Nippon Kodoshi Corporation (JP) 2014-12-24 EP disclosed
CN-104125860-A Inorganic/high molecular hybrid catalytic material with high activity in various solvents NIPPON KODOSHI CORP 2014-10-29 CN disclosed
US-20140128251-A1 INORGANIC/POLYMERIC HYBRID CATALYTIC MATERIALS CONTAINING METAL NANO-PARTICLES THEREIN NIPPON KODOSHI CORPORATION (JP) 2014-05-08 US disclosed
EP-0954375-A1 NOVEL SUPPORTED CATALYSTS Seton Hall University (US) 1999-11-10 EP disclosed
EP-0739333-B1 SELECTIVE ASYMMETRIC HYDROGENATION OF DEHYDROAMINO ACID DERIVATIVES USING RHODIUM AND IRIDIUM DIPHOSPHINITE CARBOHYDRATE CATALYST COMPOSITIONS DU PONT (US) 1998-10-14 EP disclosed
WO-1998028074-A1 NOVEL SUPPORTED CATALYSTS SETON HALL UNIVERSITY (US) 1998-07-02 WO disclosed
EP-0739333-A1 SELECTIVE ASYMMETRIC HYDROGENATION OF DEHYDROAMINO ACID DERIVATIVES USING RHODIUM AND IRIDIUM DIPHOSPHINITE CARBOHYDRATE CATALYST COMPOSITIONS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1996-10-30 EP disclosed
US-5510507-A COORDINATION CATALYSTS; EFFICIENT ENANTIOSELECTIVITY E. I. DU PONT DE NEMOURS AND COMPANY (US) 1996-04-23 US disclosed
US-5481006-A PREPARATION OF INTERMEDIATES FOR PHARMACEUTICALS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1996-01-02 US disclosed
WO-1995018787-A1 SELECTIVE ASYMMETRIC HYDROGENATION OF DEHYDROAMINO ACID DERIVATIVES USING RHODIUM AND IRIDIUM DIPHOSPHINITE CARBOHYDRATE CATALYST COMPOSITIONS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1995-07-13 WO disclosed
EP-0498507-A1 Process for the preparation of enantiomers of alpha-amino acid derivatives by asymmetric hydrogenation DSM N.V. (NL) 1992-08-12 EP disclosed