SCHEMBL23655448

SCHEMBL23655448

CC1C=CC(CC#CN)C(C(=O)O)C1

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 2/20 0.32
GRM3 Q14832 1/20 0.32
GABRR1 P24046 5/20 0.31
GABRR2 P28476 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13828461 0.75 HSD11B1 (0.34) GRM2GRM3GABRR1GABRR2
SCHEMBL284782 0.70 GABRR1 (0.36) GRM2GRM3GABRR1GABRR2
SCHEMBL27825601 0.69 GABRR1 (0.34) GRM2GRM3GABRR1GABRR2
SCHEMBL13077342 0.68 POLB (0.46) GRM2GRM3GABRR1GABRR2
Hydrochloric Acid SCHEMBL9659824 0.67 GABRR1 (0.43) GRM2GRM3GABRR1GABRR2
SCHEMBL19604954 0.65 GABRR1 (0.34) GRM2GRM3GABRR1GABRR2
SCHEMBL8926578 0.60 CYP1A2 (0.37)
SCHEMBL22133141 0.60 ABAT (0.38) GRM2GRM3GABRR1
SCHEMBL4920447 0.59
SCHEMBL1688785 0.59

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3851437-A2 METHODS OF PREPARING 1H-PYRROLO[2,3-B]PYRIDINE DERIVATES Vertex Pharmaceuticals Incorporated (US) 2021-07-21 EP disclosed