SCHEMBL2367665

SCHEMBL2367665

COc1ccc(C(C)C(=O)O)cc1N

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.57
LMNA P02545 1/20 0.57
HTT P42858 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
AKR1C3 P42330 10/20 0.55
AKR1C2 P52895 10/20 0.55
PTGS2 P35354 5/20 0.55
PTGS1 P23219 3/20 0.55
CDC42 P60953 1/20 0.55
RAC1 P63000 1/20 0.55
CYP1A2 P05177 1/20 0.55
TSHR P16473 1/20 0.55
SLC22A6 Q4U2R8 1/20 0.55
ACHE P22303 1/20 0.49
TUBB4A P04350 1/20 0.49
TUBB P07437 1/20 0.49
TUBA3C P0DPH7 1/20 0.49
TUBA1B P68363 1/20 0.49
TUBA4A P68366 1/20 0.49
TUBB4B P68371 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3315336 0.87 AKR1C3 (0.56) ALDH1A1LMNAHTTL3MBTL1AKR1C3
SCHEMBL7241661 0.85 ALDH1A1 (0.51) ALDH1A1LMNAHTTL3MBTL1PTGS2
SCHEMBL490776 0.84 ACHE (0.61) L3MBTL1AKR1C3AKR1C2PTGS2PTGS1
SCHEMBL14032691 0.84 ACHE (0.61) L3MBTL1AKR1C3AKR1C2PTGS2PTGS1
SCHEMBL5122373 0.84 ACHE (0.61) L3MBTL1AKR1C3AKR1C2PTGS2PTGS1
Hydrochloric Acid SCHEMBL3225395 0.83 ACHE (0.59) L3MBTL1AKR1C3AKR1C2PTGS2PTGS1
SCHEMBL490724 0.81 AKR1C3 (0.57) AKR1C3AKR1C2PTGS2PTGS1CDC42
SCHEMBL1002973 0.80 AKR1C3 (0.50) ALDH1A1LMNAAKR1C3AKR1C2PTGS2
SCHEMBL3667658 0.80 PTGS2 (0.61) LMNAHTTAKR1C3AKR1C2PTGS2
SCHEMBL11082037 0.80 AKR1C3 (0.55) AKR1C3AKR1C2PTGS2PTGS1CDC42

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2368887-A1 1, 2, 3-triazole derivatives for use as stearoyl-COA desaturase inhibitors Glaxosmithkline LLC (US) 2011-09-28 EP disclosed