SCHEMBL23683074

SCHEMBL23683074

C[C@H]1C=C(NC(=O)OC(C)(C)C)[C@@H](C)NC1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
GAA P10253 1/20 0.35
BRD4 O60885 2/20 0.34
CREBBP Q92793 2/20 0.34
CA1 P00915 2/20 0.33
CA2 P00918 1/20 0.33
RORC P51449 2/20 0.33
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
CYP17A1 P05093 1/20 0.32
ATR Q13535 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9438306 0.67 NFKB1 (0.34) NFKB1NFKB2RELAATR
SCHEMBL28269645 0.67 NFKB1 (0.42) EPHX2NFKB1NFKB2RELAGAA
SCHEMBL27991298 0.67 NFKB1 (0.42) EPHX2NFKB1NFKB2RELAGAA
SCHEMBL12071184 0.66 NFKB1 (0.37) EPHX2NFKB1NFKB2RELAGAA
SCHEMBL38659725 0.63 GAA (0.47) EPHX2NFKB1NFKB2RELAGAA
SCHEMBL29675032 0.63 GAA (0.45) EPHX2NFKB1NFKB2RELAGAA
SCHEMBL4317219 0.63
SCHEMBL4151983 0.63 ATR (0.39) EPHX2NFKB1NFKB2RELAGAA
SCHEMBL20689331 0.63 GAA (0.35) EPHX2NFKB1NFKB2RELAGAA
SCHEMBL13055402 0.62 CYP17A1 (0.59) GAACA1CA12CA9CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021149817-A1 Enhancement of anti-tumor activity of SHP2 inhibitor pyrimidinone in combination with novel cancer medicines in cancers TAIHO PHARMACEUTICAL CO., LTD. (JP) 2021-07-29 WO disclosed