SCHEMBL23699622

SCHEMBL23699622

Fc1ccc(-c2cc3ncn[c]c3s2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 1/20 0.50
KIT P10721 7/20 0.48
PDPK1 O15530 1/20 0.43
MAP3K8 P41279 1/20 0.43
RAB9A P51151 3/20 0.41
NPC1 O15118 2/20 0.41
MAP4K4 O95819 1/20 0.36
IKBKB O14920 2/20 0.35
CHUK O15111 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
HSD17B1 P14061 1/20 0.34
HSD17B2 P37059 1/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
FGFR1 P11362 1/20 0.34
RIPK2 O43353 1/20 0.34
STK17B O94768 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27909504 0.76 STK17B (0.36) TYK2KITRAB9ANPC1KMT2A
SCHEMBL27909495 0.76 STK17B (0.51) TYK2RAB9ANPC1KMT2ASTK17B
SCHEMBL27909505 0.76 IKBKB (0.32) IKBKBSTK17B
SCHEMBL27909499 0.76 STK17B (0.36) TYK2KITMAP3K8RAB9ANPC1
SCHEMBL27909497 0.76 HRH3 (0.44) STK17B
SCHEMBL27892406 0.74 CYP2D6 (0.47) CYP2C19
SCHEMBL27892397 0.74 IKBKB (0.31) IKBKBSTK17B
SCHEMBL28066464 0.74 EGFR (0.43)
SCHEMBL27909526 0.73 HRH3 (0.47) CYP1A2CYP3A4TDP1
SCHEMBL27909503 0.73 MAP4K4 (0.39) TYK2KITRAB9ANPC1MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2892534-B1 COMPOUNDS AND METHODS FOR KINASE MODULATION, AND INDICATIONS THEREFOR PLEXXIKON INC (US) 2021-08-04 EP disclosed