SCHEMBL27909497

SCHEMBL27909497

CCN(CC)Cc1ccc(-c2cc3ncn[c]c3s2)cc1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.44
STK17B O94768 1/20 0.36
HTR2C P28335 1/20 0.35
MCHR1 Q99705 1/20 0.35
KCNH2 Q12809 2/20 0.34
AOC3 Q16853 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27892442 0.89 AOC3 (0.35) HTR2CMCHR1KCNH2AOC3
SCHEMBL27909513 0.81 HRH3 (0.43) HRH3STK17B
SCHEMBL27909499 0.80 STK17B (0.36) STK17B
SCHEMBL27909504 0.80 STK17B (0.36) STK17B
SCHEMBL27903328 0.79 ALDH1A1 (0.42) MCHR1
SCHEMBL23699622 0.76 TYK2 (0.50) STK17B
SCHEMBL27909505 0.75 IKBKB (0.32) STK17B
SCHEMBL27909503 0.75 MAP4K4 (0.39) STK17BKCNH2
SCHEMBL28805850 0.74 CHEK1 (0.45) MCHR1KCNH2
SCHEMBL28066464 0.73 EGFR (0.43) MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102971327-A Anti-inflammatory compound having inhibitory activity against multiple tyrosine kinases, and pharmaceutical composition containing same KOREA INST SCI & TECH 2013-03-13 CN claimed
CN-102971327-B There is the anti-inflammatory compound of multiple tyrosine-kinase enzyme inhibition activity and the pharmaceutical compositions containing these compounds KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2016-04-20 CN disclosed
CN-102971327-A Anti-inflammatory compound having inhibitory activity against multiple tyrosine kinases, and pharmaceutical composition containing same KOREA INST SCI & TECH 2013-03-13 CN disclosed