SCHEMBL23709607

SCHEMBL23709607

Clc1ccc(CSc2cccc3[nH]ccc23)cc1Cl

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RHEB Q15382 6/20 0.53
PTPRG P23470 4/20 0.49
PTPRC P08575 3/20 0.41
MAPT P10636 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
HIF1A Q16665 1/20 0.41
MAOB P27338 1/20 0.41
CCR3 P51677 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5096488 0.79 RHEB (0.51) RHEBMAPTCYP1A2CYP2D6
SCHEMBL23709577 0.75 RHEB (0.71) RHEB
SCHEMBL11227010 0.71 PTPRG (0.61) PTPRGPTPRCMAPTCYP1A2CYP2D6
SCHEMBL2116708 0.71 RHEB (0.51) RHEB
SCHEMBL20535328 0.70 RHEB (1.00) RHEB
SCHEMBL23702468 0.68 RHEB (1.00) RHEBMAPT
SCHEMBL11702592 0.68 PTPRG (0.47) PTPRGPTPRCMAPTCYP1A2CYP2D6
SCHEMBL28872529 0.68 RHEB (0.76) RHEB
SCHEMBL10613968 0.67 RHEB (0.47) RHEBMAPT
Hydrochloric Acid SCHEMBL11249222 0.67 PTPRG (0.46) PTPRGPTPRCMAPTCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11339144-B2 Heteroaryl Rheb inhibitors and uses thereof NAVITOR PHARMACEUTICALS, INC. (US) 2022-05-24 US disclosed
US-20210238165-A1 HETEROARYL RHEB INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. 2021-08-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210238165-A1 HETEROARYL RHEB INHIBITORS AND USES THEREOF RHEB, KRAS, NRAS RHEB 1/4885PTPRG 2321/4885PTPRC 806/4885
US-11339144-B2 Heteroaryl Rheb inhibitors and uses thereof RHEB, GDI2, KRAS RHEB 1/4885PTPRG 3843/4885PTPRC 3141/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.