Uridine

Uridine

SCHEMBL2370972

O=P(O)(O)O.O=c1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)[nH]1.[Na].[Na]

nearest known ligand 0.88

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Uridine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC28A1 O00337 1/20 0.88
SLC28A2 O43868 1/20 0.88
SLC29A1 Q99808 1/20 0.88
SLC28A3 Q9HAS3 1/20 0.88
P2RY2 P41231 11/20 0.72
P2RY6 Q15077 8/20 0.68
P2RY4 P51582 4/20 0.67
P2RY14 Q15391 7/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Uridine SCHEMBL30094506 0.99 SLC28A1 (0.90) SLC28A1SLC28A2SLC29A1SLC28A3P2RY2
Uridine SCHEMBL29801499 0.99 SLC28A1 (0.90) SLC28A1SLC28A2SLC29A1SLC28A3P2RY2
Uridine SCHEMBL28065954 0.99 SLC28A1 (0.90) SLC28A1SLC28A2SLC29A1SLC28A3P2RY2
Uridine SCHEMBL376208 0.99 SLC28A1 (0.90) SLC28A1SLC28A2SLC29A1SLC28A3P2RY2
Uridine SCHEMBL76681 0.99 SLC28A1 (0.90) SLC28A1SLC28A2SLC29A1SLC28A3P2RY2
Uridine SCHEMBL157643 0.99 SLC28A1 (0.90) SLC28A1SLC28A2SLC29A1SLC28A3P2RY2
Uridine SCHEMBL28131489 0.97 SLC28A1 (0.88) SLC28A1SLC28A2SLC29A1SLC28A3P2RY2
Uridine SCHEMBL17074124 0.97 SLC28A1 (0.88) SLC28A1SLC28A2SLC29A1SLC28A3P2RY2
Uridine SCHEMBL29474873 0.95 SLC28A1 (0.97) SLC28A1SLC28A2SLC29A1SLC28A3P2RY2
Uridine SCHEMBL29361169 0.95 SLC28A1 (0.97) SLC28A1SLC28A2SLC29A1SLC28A3P2RY2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 59 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230293567-A1 Product and method for increasing uridine concentration in blood plasma N.V. NUTRICIA (NL) 2023-09-21 US claimed
EP-4183398-A1 COMBINATIONS OF URIDINE AND SODIUM FOR INCREASING URIDINE CONCENTRATION IN BLOOD PLASMA N.V. Nutricia (NL) 2023-05-24 EP claimed
EP-2544553-B2 CONTROLLING THE TEXTURE OF HIGH-PROTEIN NUTRITIONAL COMPOSITIONS COMPRISING MICELLAR CASEIN NUTRICIA NV (NL) 2022-11-09 EP claimed
CN-106928269-B Preparation method of phosphate 长春普华制药股份有限公司 2020-03-24 CN claimed
EP-3503899-A1 PRODUCT AND METHOD FOR INCREASING URIDINE CONCENTRATION IN BLOOD PLASMA N.V. Nutricia (NL) 2019-07-03 EP claimed
WO-2018038599-A1 PRODUCT AND METHOD FOR INCREASING URIDINE CONCENTRATION IN BLOOD PLASMA N.V. NUTRICIA (NL) 2018-03-01 WO claimed
WO-2018038609-A1 PRODUCT AND METHOD FOR INCREASING URIDINE CONCENTRATION IN BLOOD PLASMA N.V. NUTRICIA (NL) 2018-03-01 WO claimed
US-9872888-B2 Use of a nucleotide for improving the heat stability of an aqueous micellar casein composition N.V. NUTRICIA (NL) 2018-01-23 US claimed
EP-2732710-B1 Controlling the texture of high-protein nutritional compositions comprising micellar casein NUTRICIA NV (NL) 2015-07-29 EP claimed
EP-2734060-A1 USE OF A NUCLEOTIDE FOR IMPROVING THE HEAT STABILITY OF AN AQUEOUS MICELLAR CASEIN COMPOSITION N.V. Nutricia (NL) 2014-05-28 EP claimed
EP-2732710-A1 Controlling the texture of high-protein nutritional compositions comprising micellar casein N.V. Nutricia (NL) 2014-05-21 EP claimed
US-20140135257-A1 USE OF A NUCLEOTIDE FOR IMPROVING THE HEAT STABILITY OF AN AQUEOUS MICELLAR CASEIN COMPOSITION N.V. NUTRICIA 2014-05-15 US claimed
EP-2544553-B1 CONTROLLING THE TEXTURE OF HIGH-PROTEIN NUTRITIONAL COMPOSITIONS COMPRISING MICELLAR CASEIN NUTRICIA NV (NL) 2014-02-26 EP claimed
US-20130065824-A1 CONTROLLING THE TEXTURE OF HIGH-PROTEIN NUTRITIONAL COMPOSITIONS COMPRISING MICELLAR CASEIN N.V. NUTRICIA 2013-03-14 US claimed
WO-2013012313-A1 USE OF A NUCLEOTIDE FOR IMPROVING THE HEAT STABILITY OF AN AQUEOUS MICELLAR CASEIN COMPOSITION N.V. NUTRICIA (NL) 2013-01-24 WO claimed
WO-2013012324-A1 USE OF A NUCLEOTIDE FOR IMPROVING THE HEAT STABILITY OF AN AQUEOUS MICELLAR CASEIN COMPOSITION N.V. NUTRICIA (NL) 2013-01-24 WO claimed
EP-2544553-A1 CONTROLLING THE TEXTURE OF HIGH-PROTEIN NUTRITIONAL COMPOSITIONS COMPRISING MICELLAR CASEIN N.V. Nutricia (NL) 2013-01-16 EP claimed
WO-2011112075-A1 CONTROLLING THE TEXTURE OF HIGH-PROTEIN NUTRITIONAL COMPOSITIONS COMPRISING MICELLAR CASEIN N.V. NUTRICIA (NL) 2011-09-15 WO claimed
WO-2011112087-A1 CONTROLLING THE TEXTURE OF HIGH-PROTEIN NUTRITIONAL COMPOSITIONS COMPRISING MICELLAR CASEIN N.V. NUTRICIA (NL) 2011-09-15 WO claimed
EP-4353261-A1 NUTRACEUTIC COMBINATION AND ITS USE IN THE TREATMENT OF NEUROLOGICAL DISORDERS Hospital Sant Joan de Deu (ES) 2024-04-17 EP disclosed
CN-113784706-B Multi-layered pharmaceutical or nutraceutical solid dosage forms comprising pyrimidine and/or purine derivatives and B vitamins, their preparation and use 菲尔若国际公司 2024-01-05 CN disclosed
US-20240000124-A1 DAIRY PRODUCT AND PROCESS FONTERRA COOPERATIVE GROUP LTD (NZ) 2024-01-04 US disclosed
US-20230293567-A1 Product and method for increasing uridine concentration in blood plasma N.V. NUTRICIA (NL) 2023-09-21 US disclosed
CN-116768948-A Method for synthesizing urine phosphorylcholine in citicoline injection 山东玉满坤生物科技有限公司 2023-09-19 CN disclosed
CN-116768948-A Method for synthesizing urine phosphorylcholine in citicoline injection 山东玉满坤生物科技有限公司 2023-09-19 CN disclosed
EP-4228417-A1 DAIRY PRODUCT AND PROCESS Fonterra Co-Operative Group Limited (NZ) 2023-08-23 EP disclosed
US-11707478-B2 Method for increasing uridine concentration in blood plasma N.V. NUTRICIA (NL) 2023-07-25 US disclosed
CN-116284187-A Method for synthesizing urine phosphorylcholine in citicoline injection 山东玉满坤生物科技有限公司 2023-06-23 CN disclosed
EP-4183398-A1 COMBINATIONS OF URIDINE AND SODIUM FOR INCREASING URIDINE CONCENTRATION IN BLOOD PLASMA N.V. Nutricia (NL) 2023-05-24 EP disclosed
CN-115916151-A Expanded foams for delivery of functional ingredients 勃林格殷格翰动物保健有限公司 2023-04-04 CN disclosed
EP-3503899-B1 PRODUCT AND METHOD FOR INCREASING URIDINE CONCENTRATION IN BLOOD PLASMA NUTRICIA NV (NL) 2022-11-23 EP disclosed
EP-2544553-B2 CONTROLLING THE TEXTURE OF HIGH-PROTEIN NUTRITIONAL COMPOSITIONS COMPRISING MICELLAR CASEIN NUTRICIA NV (NL) 2022-11-09 EP disclosed
CN-111662350-B Preparation method of green intelligent high-purity diquafosol tetrasodium 南京宸翔医药研究有限责任公司 2022-06-07 CN disclosed
CN-111662350-B Preparation method of green intelligent high-purity diquafosol tetrasodium 南京宸翔医药研究有限责任公司 2022-06-07 CN disclosed
CN-109789161-B Products and methods for increasing uridine concentration in plasma N·V·努特里奇亚 2022-04-22 CN disclosed
WO-2022079673-A1 DAIRY PRODUCT AND PROCESS FONTERRA CO-OPERATIVE GROUP LIMITED (NZ) 2022-04-21 WO disclosed
CN-111662350-A Preparation method of green intelligent high-purity diquafosol tetrasodium 南京宸翔医药研究有限责任公司 2020-09-15 CN disclosed
CN-111662350-A Preparation method of green intelligent high-purity diquafosol tetrasodium 南京宸翔医药研究有限责任公司 2020-09-15 CN disclosed
CN-110944622-A External composition 大塚制药株式会社 2020-03-31 CN disclosed
EP-3503899-A1 PRODUCT AND METHOD FOR INCREASING URIDINE CONCENTRATION IN BLOOD PLASMA N.V. Nutricia (NL) 2019-07-03 EP disclosed
US-20190183916-A1 PRODUCT AND METHOD FOR INCREASING URIDINE CONCENTRATION IN BLOOD PLASMA N.V. NUTRICIA (NL) 2019-06-20 US disclosed
US-10264806-B2 Controlling the texture of high-protein nutritional compositions comprising micellar casein N.V. NUTRICIA (NL) 2019-04-23 US disclosed
WO-2018038599-A1 PRODUCT AND METHOD FOR INCREASING URIDINE CONCENTRATION IN BLOOD PLASMA N.V. NUTRICIA (NL) 2018-03-01 WO disclosed
WO-2018038609-A1 PRODUCT AND METHOD FOR INCREASING URIDINE CONCENTRATION IN BLOOD PLASMA N.V. NUTRICIA (NL) 2018-03-01 WO disclosed
US-9872888-B2 Use of a nucleotide for improving the heat stability of an aqueous micellar casein composition N.V. NUTRICIA (NL) 2018-01-23 US disclosed
EP-2734060-B1 USE OF A NUCLEOTIDE FOR IMPROVING THE HEAT STABILITY OF AN AQUEOUS MICELLAR CASEIN COMPOSITION NUTRICIA NV (NL) 2017-11-29 EP disclosed
EP-2732710-B1 Controlling the texture of high-protein nutritional compositions comprising micellar casein NUTRICIA NV (NL) 2015-07-29 EP disclosed
EP-2734060-A1 USE OF A NUCLEOTIDE FOR IMPROVING THE HEAT STABILITY OF AN AQUEOUS MICELLAR CASEIN COMPOSITION N.V. Nutricia (NL) 2014-05-28 EP disclosed
EP-2732710-A1 Controlling the texture of high-protein nutritional compositions comprising micellar casein N.V. Nutricia (NL) 2014-05-21 EP disclosed
US-20140135257-A1 USE OF A NUCLEOTIDE FOR IMPROVING THE HEAT STABILITY OF AN AQUEOUS MICELLAR CASEIN COMPOSITION N.V. NUTRICIA 2014-05-15 US disclosed
EP-2544553-B1 CONTROLLING THE TEXTURE OF HIGH-PROTEIN NUTRITIONAL COMPOSITIONS COMPRISING MICELLAR CASEIN NUTRICIA NV (NL) 2014-02-26 EP disclosed
US-20130065824-A1 CONTROLLING THE TEXTURE OF HIGH-PROTEIN NUTRITIONAL COMPOSITIONS COMPRISING MICELLAR CASEIN N.V. NUTRICIA 2013-03-14 US disclosed
WO-2013012313-A1 USE OF A NUCLEOTIDE FOR IMPROVING THE HEAT STABILITY OF AN AQUEOUS MICELLAR CASEIN COMPOSITION N.V. NUTRICIA (NL) 2013-01-24 WO disclosed
WO-2013012324-A1 USE OF A NUCLEOTIDE FOR IMPROVING THE HEAT STABILITY OF AN AQUEOUS MICELLAR CASEIN COMPOSITION N.V. NUTRICIA (NL) 2013-01-24 WO disclosed
EP-2544553-A1 CONTROLLING THE TEXTURE OF HIGH-PROTEIN NUTRITIONAL COMPOSITIONS COMPRISING MICELLAR CASEIN N.V. Nutricia (NL) 2013-01-16 EP disclosed
WO-2011112075-A1 CONTROLLING THE TEXTURE OF HIGH-PROTEIN NUTRITIONAL COMPOSITIONS COMPRISING MICELLAR CASEIN N.V. NUTRICIA (NL) 2011-09-15 WO disclosed
WO-2011112087-A1 CONTROLLING THE TEXTURE OF HIGH-PROTEIN NUTRITIONAL COMPOSITIONS COMPRISING MICELLAR CASEIN N.V. NUTRICIA (NL) 2011-09-15 WO disclosed
US-6194009-B1 INSTANT FOODS; LINOLEIC AND LINOLENIC ACIDS; NUTRITIONALLY BALANCED PRINCETON NUTRITION, LLC 2001-02-27 US disclosed
WO-1998006277-A1 NUTRITIONAL FORMULAS SUPPLEMENTED WITH NUCLEOTIDES, AND PROCESSES THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 1998-02-19 WO disclosed
WO-1998006277-A1 NUTRITIONAL FORMULAS SUPPLEMENTED WITH NUCLEOTIDES, AND PROCESSES THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 1998-02-19 WO disclosed