SCHEMBL23715797

SCHEMBL23715797

N=C(NC(O)C(NNOc1ccc(Cl)c(Cl)c1)C1CCOCC1)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 15/20 0.35
S1PR4 O95977 8/20 0.33
S1PR1 P21453 3/20 0.33
S1PR5 Q9H228 3/20 0.33
S1PR2 O95136 2/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
KMO O15229 1/20 0.30
HRH1 P35367 1/20 0.30
CCR3 P51677 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23715847 0.73 S1PR3 (0.42) S1PR3S1PR4S1PR1S1PR5S1PR2
SCHEMBL23715831 0.71 S1PR3 (0.47) S1PR3S1PR4S1PR1S1PR5S1PR2
SCHEMBL23716419 0.70 SLC6A3 (0.35) KCNH2
SCHEMBL23715838 0.69 S1PR3 (0.45) S1PR3S1PR4S1PR1S1PR5S1PR2
SCHEMBL23716190 0.68 SLC6A3 (0.41) NPSR1
SCHEMBL17663846 0.67 S1PR3 (0.61) S1PR3S1PR4S1PR1S1PR5S1PR2
SCHEMBL23716102 0.65 S1PR3 (0.40) S1PR3S1PR4S1PR1S1PR5S1PR2
SCHEMBL23715998 0.64 S1PR3 (0.42) S1PR3S1PR4S1PR1S1PR5S1PR2
SCHEMBL23715785 0.62 S1PR3 (0.48) S1PR3S1PR4S1PR1S1PR5CYP3A4
SCHEMBL17663806 0.61 NPC1 (0.45) S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3209732-B1 SPHINGOSINE-1-PHOSPATE RECEPTOR MODULATORS FOR TREATMENT OF CARDIOPULMONARY DISORDERS SCRIPPS RESEARCH INST (US) 2021-08-04 EP disclosed