SCHEMBL23716100

SCHEMBL23716100

NC(c1ccc(Cl)cc1)c1ccc(Cl)nc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 2/20 0.45
S1PR1 P21453 1/20 0.45
ADRB2 P07550 1/20 0.43
AKT2 P31751 1/20 0.41
CYP19A1 P11511 3/20 0.38
PIK3CD O00329 1/20 0.38
KCNQ3 O43525 1/20 0.38
KCNQ2 O43526 1/20 0.38
KCNE1 P15382 1/20 0.38
KCNQ1 P51787 1/20 0.38
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
ADRA2A P08913 2/20 0.36
ADRA2B P18089 2/20 0.36
ADRA2C P18825 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3382818 0.86 CYP3A4 (0.42) AKT2PIK3CDKCNQ3KCNQ2CYP3A4
SCHEMBL1732927 0.80 ADRB2 (0.62) S1PR3S1PR1ADRB2AKT2CYP19A1
SCHEMBL11538507 0.79 CYP19A1 (0.55) S1PR3ADRB2CYP19A1PIK3CDKCNQ3
SCHEMBL13567642 0.79 PIK3CD (0.43) ADRB2PIK3CDCYP3A4CYP2D6SLC6A2
SCHEMBL3828644 0.79 PIK3CD (0.43) ADRB2PIK3CDCYP3A4CYP2D6SLC6A2
SCHEMBL4165718 0.79 PIK3CD (0.43) ADRB2PIK3CDCYP3A4CYP2D6SLC6A2
Hydrochloric Acid SCHEMBL3179658 0.78 ADRB2 (0.59) S1PR3S1PR1ADRB2AKT2CYP19A1
SCHEMBL3299158 0.76 KCNQ3 (0.41) S1PR3CYP19A1KCNQ3KCNQ2KCNE1
SCHEMBL3297715 0.76 CYP19A1 (0.38) S1PR3S1PR1ADRB2CYP19A1PIK3CD
SCHEMBL6420457 0.76 CYP3A4 (0.39) S1PR3S1PR1AKT2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3209732-B1 SPHINGOSINE-1-PHOSPATE RECEPTOR MODULATORS FOR TREATMENT OF CARDIOPULMONARY DISORDERS SCRIPPS RESEARCH INST (US) 2021-08-04 EP disclosed