SCHEMBL2371728

SCHEMBL2371728

COc1ccc2c(c1)C1(CNC[C@H](N)O1)c1cc(Br)ccc1O2

nearest known ligand 0.37

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 14/20 0.36
CTSD P07339 7/20 0.34
SIRT2 Q8IXJ6 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2370894 1.00 BACE1 (0.36) BACE1CTSDSIRT2
SCHEMBL2370832 0.87 BACE1 (0.35) BACE1
SCHEMBL2371098 0.87 BACE1 (0.35) BACE1
SCHEMBL2371315 0.87 BACE1 (0.35) BACE1CTSD
SCHEMBL2371365 0.87 BACE1 (0.35) BACE1
SCHEMBL2371275 0.84 BACE1 (0.37) BACE1
SCHEMBL2370327 0.83 BACE1 (0.32) BACE1
SCHEMBL2370741 0.83 OPRM1 (0.33) BACE1
SCHEMBL2370531 0.79 BACE1 (0.50) BACE1CTSD
SCHEMBL2370410 0.79 BACE1 (0.50) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2547686-A1 AMINO -DIHYDROOXAZINE AND AMINO - DIHYDROTHIAZINE SPIRO COMPOUNDS AS BETA - SECRETASE MODULATORS AND THEIR MEDICAL USE Amgen Inc. (US) 2013-01-23 EP disclosed
WO-2011115928-A1 AMINO -DIHYDROOXAZINE AND AMINO - DIHYDROTHIAZINE SPIRO COMPOUNDS AS BETA - SECRETASE MODULATORS AND THEIR MEDICAL USE AMGEN INC. (US) 2011-09-22 WO disclosed