SCHEMBL23719010

SCHEMBL23719010

CN(C)C1(c2ccccc2)CCN(C(=O)[C@H]2Cc3ccccc3CN2)CC1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.48
ROCK2 O75116 1/20 0.47
CYP3A4 P08684 1/20 0.47
ARG1 P05089 1/20 0.44
ARG2 P78540 1/20 0.44
OPRL1 P41146 15/20 0.44
OPRM1 P35372 10/20 0.44
OPRK1 P41145 2/20 0.42
SMYD3 Q9H7B4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23719118 1.00 KMT2A (0.48) KMT2AROCK2CYP3A4ARG1ARG2
SCHEMBL23719120 1.00 KMT2A (0.48) KMT2AROCK2CYP3A4ARG1ARG2
Hydrochloric Acid SCHEMBL23699217 0.99 KMT2A (0.48) KMT2AROCK2CYP3A4ARG1ARG2
Hydrochloric Acid SCHEMBL23699215 0.99 KMT2A (0.48) KMT2AROCK2CYP3A4ARG1ARG2
Hydrochloric Acid SCHEMBL23699268 0.99 KMT2A (0.48) KMT2AROCK2CYP3A4ARG1ARG2
SCHEMBL23719083 0.83 OPRL1 (0.41) OPRL1OPRM1OPRK1
SCHEMBL25375448 0.82 ROCK2 (0.52) KMT2AROCK2CYP3A4ARG1ARG2
SCHEMBL31263918 0.82 ROCK2 (0.52) KMT2AROCK2CYP3A4ARG1ARG2
SCHEMBL25377868 0.82 ROCK2 (0.52) KMT2AROCK2CYP3A4ARG1ARG2
Hydrochloric Acid SCHEMBL23699334 0.82 OPRL1 (0.41) OPRL1OPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3858439-A1 AMIDE DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN ESTEVE PHARMACEUTICALS, S.A. (ES) 2021-08-04 EP disclosed