SCHEMBL23724890

SCHEMBL23724890

COc1nc(-c2cccc(Br)c2Cl)ccc1CN(CC1CCC(=O)N1)C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 20/20 0.57
PDCD1LG2 Q9BQ51 17/20 0.57
PDCD1 Q15116 3/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25175600 1.00 CD274 (0.57) CD274PDCD1LG2PDCD1
SCHEMBL25172047 0.98 CD274 (0.60) CD274PDCD1LG2PDCD1
SCHEMBL23727030 0.98 CD274 (0.60) CD274PDCD1LG2PDCD1
SCHEMBL21496984 0.92 CD274 (0.56) CD274PDCD1LG2PDCD1
SCHEMBL23725822 0.90 CD274 (0.54) CD274PDCD1LG2PDCD1
SCHEMBL23726118 0.89 CD274 (0.56) CD274PDCD1LG2PDCD1
SCHEMBL23725246 0.88 PDCD1 (0.70) CD274PDCD1
SCHEMBL23725217 0.87 PDCD1LG2 (0.60) CD274PDCD1LG2
SCHEMBL25169163 0.87 PDCD1LG2 (0.60) CD274PDCD1LG2
SCHEMBL27080091 0.87 CD274 (0.58) CD274PDCD1LG2PDCD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4313968-A2 SUBSTITUTED 1-ARYL-1'-HETEROARYL COMPOUNDS, SUBSTITUTED 1,1'-BIHETEROARYL COMPOUNDS, AND METHODS USING SAME Arbutus Biopharma Corporation (CA) 2024-02-07 EP disclosed
US-20230143612-A1 SUBSTITUTED 1,1'-BIPHENYL COMPOUNDS AND METHODS USING SAME ARBUTUS BIOPHARMA CORP (US) 2023-05-11 US disclosed
EP-4100381-A1 SUBSTITUTED 1,1'-BIPHENYL COMPOUNDS AND METHODS USING SAME Arbutus Biopharma Corporation (CA) 2022-12-14 EP disclosed
WO-2021158481-A1 SUBSTITUTED 1,1'-BIPHENYL COMPOUNDS AND METHODS USING SAME ARBUTUS BIOPHARMA, INC. (US) 2021-08-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230143612-A1 SUBSTITUTED 1,1'-BIPHENYL COMPOUNDS AND METHODS USING SAME HAVCR2, HMBS, VHL CD274 75/4885PDCD1LG2 225/4885PDCD1 62/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.