SCHEMBL23730433

SCHEMBL23730433

CCC(CC)Oc1cc2c(Nc3ccc(C(F)(F)F)cc3)c(C#N)cnc2cc1OC

nearest known ligand 0.67

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.67
ERBB2 P04626 7/20 0.67
MAP2K1 Q02750 7/20 0.63
SRC P12931 5/20 0.62
RAF1 P04049 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6380567 0.91 EGFR (0.79) EGFRERBB2MAP2K1SRCRAF1
SCHEMBL23730429 0.85 SRC (0.64) EGFRERBB2SRC
SCHEMBL6381464 0.81 EGFR (1.00) EGFRERBB2MAP2K1SRCRAF1
SCHEMBL6381317 0.80 EGFR (1.00) EGFRERBB2MAP2K1SRCRAF1
SCHEMBL6382822 0.79 MAP2K1 (0.78) EGFRERBB2MAP2K1SRCRAF1
SCHEMBL23730140 0.79 EGFR (0.62) EGFRERBB2MAP2K1SRCRAF1
SCHEMBL6381609 0.78 EGFR (1.00) EGFRERBB2MAP2K1SRCRAF1
SCHEMBL5733290 0.77 MAP2K1 (1.00) EGFRERBB2MAP2K1SRCRAF1
SCHEMBL6380423 0.77 EGFR (1.00) EGFRERBB2MAP2K1SRC
SCHEMBL28756490 0.77 MAP2K1 (0.95) EGFRERBB2MAP2K1SRCRAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021155144-A1 USE OF QUINAZOLINE-BASED TYROSINE KINASE INHIBITORS FOR THE TREATMENT OF CANCERS WITH NRG1 FUSIONS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2021-08-05 WO disclosed