SCHEMBL23733453

SCHEMBL23733453

CCN[C@H](CCO)C(=O)N1CCc2nc(C(C)C)ccc2C1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 9/20 0.36
ACE P12821 2/20 0.34
KCNH2 Q12809 3/20 0.34
HSP90B1 P14625 3/20 0.34
GPBAR1 Q8TDU6 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 1/20 0.33
MMP1 P03956 1/20 0.33
MMP3 P08254 1/20 0.33
MMP9 P14780 1/20 0.33
KMT2A Q03164 1/20 0.33
MAPK1 P28482 1/20 0.33
FPR2 P25090 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20203495 0.79 ACE (0.40) HSP90AA1ACEHSP90B1
SCHEMBL18806180 0.78 CDK1 (0.44) HSP90AA1KCNH2HSP90B1GPBAR1KDM4E
SCHEMBL18819907 0.75 HSP90AA1 (0.38) HSP90AA1HSP90B1
SCHEMBL20203602 0.72 CDK1 (0.41) HSP90AA1KDM4EALDH1A1KMT2A
SCHEMBL20203582 0.71 KDR (0.40) HSP90AA1KDM4EALDH1A1
SCHEMBL23733468 0.71 NPC1 (0.42) HSP90AA1KDM4EALDH1A1
SCHEMBL20203643 0.71 HSP90AA1 (0.40) HSP90AA1KCNH2HSP90B1
SCHEMBL20203586 0.71 ALDH1A1 (0.37) HSP90AA1HSP90B1KDM4EALDH1A1KMT2A
SCHEMBL20203456 0.71 GRM5 (0.41) HSP90AA1KCNH2ALDH1A1TP53KMT2A
SCHEMBL23733491 0.70 CYP2C19 (0.38) HSP90AA1KCNH2HSP90B1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11084814-B2 Pyrido[3, 4-d]pyrimidine derivative and pharmaceutically acceptable salt thereof TEIJIN PHARMA LIMITED (JP) 2021-08-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11084814-B2 Pyrido[3, 4-d]pyrimidine derivative and pharmaceutically acceptable salt thereof CDK4, CDK6, CDK16 HSP90AA1 4289/4885ACE 404/4885KCNH2 3188/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.