SCHEMBL23733474

SCHEMBL23733474

CC(C)c1ccc2c(n1)CCN(C(=O)C1CCCN1)C2

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 2/20 0.45
CDK4 P11802 2/20 0.45
CDK2 P24941 2/20 0.45
CDK7 P50613 2/20 0.45
CDK9 P50750 2/20 0.45
CDK6 Q00534 2/20 0.45
PARP1 P09874 1/20 0.44
P2RX7 Q99572 1/20 0.39
CGAS Q8N884 1/20 0.39
DPP4 P27487 1/20 0.38
DPP8 Q6V1X1 1/20 0.38
DPP9 Q86TI2 1/20 0.38
HSP90AA1 P07900 7/20 0.38
HSP90B1 P14625 1/20 0.37
CCR4 P51679 1/20 0.37
PIK3CD O00329 2/20 0.35
PIK3CA P42336 2/20 0.35
PIK3CB P42338 2/20 0.35
PIK3CG P48736 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20203529 1.00 CDK1 (0.45) CDK1CDK4CDK2CDK7CDK9
SCHEMBL23733478 0.97 CDK1 (0.43) CDK1CDK4CDK2CDK7CDK9
SCHEMBL20203569 0.94 CDK1 (0.40) CDK1CDK4CDK2CDK7CDK9
SCHEMBL23733451 0.83 KEAP1 (0.40) PARP1HSP90AA1
SCHEMBL20203431 0.82 KEAP1 (0.41) CDK1CDK4HSP90AA1HSP90B1
SCHEMBL23733475 0.82 DPP4 (0.39) CDK4CDK2CDK6DPP4DPP8
SCHEMBL20203568 0.82 DPP4 (0.39) CDK4CDK2CDK6DPP4DPP8
SCHEMBL20203531 0.80 TLR9 (0.41) CDK1CDK4CDK2CDK6PARP1
SCHEMBL20203457 0.80 GRM5 (0.49) CDK1CDK4HSP90AA1
SCHEMBL23733477 0.80 CDK1 (0.45) CDK1CDK4CDK2CDK7CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11084814-B2 Pyrido[3, 4-d]pyrimidine derivative and pharmaceutically acceptable salt thereof TEIJIN PHARMA LIMITED (JP) 2021-08-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11084814-B2 Pyrido[3, 4-d]pyrimidine derivative and pharmaceutically acceptable salt thereof CDK4, CDK6, CDK16 CDK1 8/4885CDK4 1/4885CDK2 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.