SCHEMBL23744329

SCHEMBL23744329

CN(C)C(=O)c1cnc(N2CCNCC2)nc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.53
CLK4 Q9HAZ1 2/20 0.53
CYP2D6 P10635 2/20 0.53
HSD17B10 Q99714 4/20 0.47
USP2 O75604 2/20 0.47
HDAC6 Q9UBN7 2/20 0.46
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 1/20 0.46
OPRD1 P41143 1/20 0.44
TAAR1 Q96RJ0 1/20 0.43
DGAT2 Q96PD7 1/20 0.43
POLB P06746 1/20 0.43
CYP1A2 P05177 4/20 0.40
CASP1 P29466 3/20 0.40
CASP7 P55210 3/20 0.40
CYP3A4 P08684 2/20 0.40
HPGD P15428 2/20 0.40
CYP2C19 P33261 2/20 0.40
OPRM1 P35372 1/20 0.39
OPRL1 P41146 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16651634 0.82 ALDH1A1 (0.50) TSHRCLK4CYP2D6HSD17B10USP2
SCHEMBL27507507 0.82 HDAC6 (0.44) TSHRCLK4CYP2D6HSD17B10USP2
SCHEMBL15286548 0.81 TSHR (0.56) TSHRCLK4CYP2D6HSD17B10USP2
SCHEMBL598464 0.80 POLB (0.65) TSHRHSD17B10USP2HDAC6ALDH1A1
SCHEMBL25419798 0.79 CHRNB2 (0.51) TSHRHSD17B10HDAC6ALDH1A1KDM4E
SCHEMBL12485764 0.79 TAAR1 (0.51) TSHRCLK4CYP2D6HSD17B10USP2
SCHEMBL3613525 0.78 OGA (0.49) TSHRHSD17B10HDAC6ALDH1A1KDM4E
SCHEMBL23560975 0.78 HDAC6 (0.55) TSHRHSD17B10HDAC6ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL30422704 0.78 ALDH1A1 (0.53) TSHRHSD17B10HDAC6ALDH1A1KDM4E
SCHEMBL23064392 0.77 TSHR (0.53) TSHRCLK4CYP2D6HSD17B10USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021158698-A1 MUSCARINIC RECEPTOR 4 ANTAGONISTS AND METHODS OF USE NEUROCRINE BIOSCIENCES, INC. (US) 2021-08-12 WO disclosed