SCHEMBL23747152

SCHEMBL23747152

O=C(Nc1ncnn2c(Br)ccc12)NC1CC1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.41
HTR3A P46098 1/20 0.41
KCNH2 Q12809 1/20 0.41
SIGMAR1 Q99720 5/20 0.40
HTT P42858 2/20 0.39
EPHX1 P07099 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
AURKA O14965 1/20 0.36
AURKB Q96GD4 1/20 0.36
TTK P33981 1/20 0.36
GAA P10253 1/20 0.36
PAK1 Q13153 1/20 0.35
KDR P35968 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
EPHX2 P34913 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23746987 0.85 KDR (0.45) CHRNA7HTR3ASIGMAR1HTTEPHX1
SCHEMBL23747016 0.69 CHRNA7 (0.41) CHRNA7HTR3AKCNH2
SCHEMBL23747109 0.68 CHRNA7 (0.41) CHRNA7HTR3AKCNH2HTTMEN1
SCHEMBL21199010 0.67 MAPT (0.44) CHRNA7HTR3AKCNH2HTTMEN1
SCHEMBL23747030 0.65 FKBP1A (0.43) CHRNA7HTR3AKCNH2HTTMEN1
SCHEMBL25219260 0.64 CHRNA7 (0.38) CHRNA7HTR3AKCNH2KDR
SCHEMBL23747015 0.63 CCR4 (0.42) MEN1KMT2AAURKBSMN1; SMN2
SCHEMBL4047301 0.63 KDR (0.51) CHRNA7HTR3AKCNH2HTTMEN1
SCHEMBL23747216 0.62 EDNRB (0.40) CHRNA7HTR3AKCNH2HTTMEN1
SCHEMBL23747116 0.62 CHRNA7 (0.35) CHRNA7HTR3AKCNH2TTKKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021158516-A1 IRE1α MODULATORS AND USES THEREOF NIMBUS IASO, INC. (US) 2021-08-12 WO disclosed