SCHEMBL23747016

SCHEMBL23747016

O=S(=O)(Nc1ncnn2c(Br)ccc12)C1CCCC1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.41
HTR3A P46098 2/20 0.41
KCNH2 Q12809 1/20 0.41
BRPF1 P55201 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
EGLN2 Q96KS0 1/20 0.34
BRAF P15056 1/20 0.31
FPR1 P21462 1/20 0.31
SGK1 O00141 1/20 0.30
PIP4K2A P48426 1/20 0.30
PIK3CA P42336 1/20 0.30
BRD4 O60885 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23747109 0.99 CHRNA7 (0.41) CHRNA7HTR3AKCNH2BRPF1TDP1
SCHEMBL23746997 0.85 EGFR (0.43) CHRNA7HTR3ABRPF1TDP1EGLN2
SCHEMBL23746999 0.84 EGFR (0.42) CHRNA7HTR3ABRPF1EGLN2BRAF
SCHEMBL23747030 0.78 FKBP1A (0.43) CHRNA7HTR3AKCNH2
SCHEMBL23747015 0.74 CCR4 (0.42) EGLN2
SCHEMBL23747216 0.73 EDNRB (0.40) CHRNA7HTR3AKCNH2BRAF
SCHEMBL23747082 0.70 CCR4 (0.46)
SCHEMBL23747149 0.70 PTGS1 (0.35) CHRNA7HTR3AKCNH2BRAF
SCHEMBL23747096 0.70 EDNRA (0.42) TDP1SGK1
SCHEMBL23747152 0.69 CHRNA7 (0.41) CHRNA7HTR3AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021158516-A1 IRE1α MODULATORS AND USES THEREOF NIMBUS IASO, INC. (US) 2021-08-12 WO disclosed