SCHEMBL23747737

SCHEMBL23747737

O=C(NCc1ccc(Cl)cc1)Nc1ccc(S(=O)(=O)Nc2ccnn2-c2ccccc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 10/20 0.61
KMT2A Q03164 2/20 0.61
CYP2C9 P11712 6/20 0.56
CYP2C8 P10632 1/20 0.56
OXTR P30559 2/20 0.54
CYP2C19 P33261 2/20 0.53
LMNA P02545 1/20 0.53
POLB P06746 1/20 0.53
CYP3A4 P08684 1/20 0.53
TSHR P16473 1/20 0.53
NFKB1 P19838 1/20 0.53
CYP2C18 P33260 1/20 0.53
THPO P40225 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
HSD17B10 Q99714 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
KDM4E B2RXH2 1/20 0.51
MEN1 O00255 1/20 0.51
MAPT P10636 1/20 0.51
AVPR1A P37288 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12335073 0.78 NAMPT (0.93) NAMPT
SCHEMBL17325743 0.76 NAMPT (1.00) NAMPT
SCHEMBL8551429 0.76 CYP2C9 (0.56) KMT2ACYP2C9CYP2C8OXTRCYP2C19
SCHEMBL20379304 0.76 NAMPT (1.00) NAMPT
SCHEMBL6199073 0.76 CYP2C9 (0.47) KMT2ACYP2C9CYP2C8OXTRCYP2C19
SCHEMBL23727738 0.74 NAMPT (0.72) NAMPTKMT2APOLBKDM4EMEN1
SCHEMBL23747550 0.73 NAMPT (0.73) NAMPTKMT2APOLBMEN1MAPT
SCHEMBL20379216 0.73 NAMPT (1.00) NAMPT
SCHEMBL20379606 0.73 NAMPT (1.00) NAMPT
SCHEMBL3849178 0.73 CYP2C9 (0.71) KMT2ACYP2C9CYP2C8OXTRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230133132-A1 NAMPT MODULATORS CYTOKINETICS, INC. 2023-05-04 US disclosed
US-20230133132-A1 NAMPT MODULATORS CYTOKINETICS, INC. 2023-05-04 US disclosed
US-20230133132-A1 NAMPT MODULATORS CYTOKINETICS, INC. 2023-05-04 US disclosed
WO-2021159015-A1 NAMPT MODULATORS CYTOKINETICS, INC. (US) 2021-08-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230133132-A1 NAMPT MODULATORS NAMPT, MC4R, SIRT1 NAMPT 1/4885KMT2A 1669/4885CYP2C9 1927/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.