SCHEMBL237495

SCHEMBL237495

CC(C)(C)C(COC(N)=O)c1cccc(C#CCCCO)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
EGFR P00533 1/20 0.37
CYP1A2 P05177 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
CYP2D6 P10635 1/20 0.36
PKM P14618 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
BACE1 P56817 1/20 0.34
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA5 P31644 1/20 0.33
GABRA3 P34903 1/20 0.33
GABRA2 P47869 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4178359 0.78 HTR2C (0.39) HTR2CHTR2BEGFRCYP1A2CHRNB4
SCHEMBL3879268 0.77 BACE1 (0.35) CYP1A2SMN1; SMN2CYP2D6PKMNPSR1
SCHEMBL237494 0.74 HTR2C (0.38) HTR2CHTR2BEGFRCHRNB4CHRNA3
SCHEMBL28432379 0.73 CYP1A2 (0.62) CYP1A2SMN1; SMN2CYP2D6PKMNPSR1
SCHEMBL4178362 0.72 LMNA (0.47) HTR2CHTR2BEGFRCHRNB4CHRNA3
SCHEMBL237493 0.72 HTR2C (0.40) HTR2CHTR2BEGFRCHRNB4CHRNA3
SCHEMBL27807256 0.70 ACACB (0.42) HTR2CHTR2BEGFRCHRNB4CHRNA3
SCHEMBL2180350 0.69 HTR2C (0.51) HTR2CHTR2BEGFRCYP1A2CHRNB4
SCHEMBL236187 0.69 ALDH1A1 (0.37) CYP1A2ALDH1A1CYP3A4MAPTCYP2C9
SCHEMBL236559 0.68 HTR2C (0.44) HTR2CHTR2BEGFRCYP1A2CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120004269-A1 Alkynyl Phenyl Derivative Compounds for Treating Ophthalmic Diseases and Disorders ACUCELA INC. (US) 2012-01-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120004269-A1 Alkynyl Phenyl Derivative Compounds for Treating Ophthalmic Diseases and Disorders PDE6D, STARD3, PDE6C HTR2C 3284/4885HTR2B 2548/4885EGFR 1703/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.