SCHEMBL23749523

SCHEMBL23749523

Nc1ccc(Oc2ncnc3cc(OCCCN4CCOCC4)c4c(c23)OCCO4)c(F)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 5/20 0.64
RAF1 P04049 4/20 0.64
KDR P35968 10/20 0.63
EGFR P00533 6/20 0.59
AXL P30530 2/20 0.57
RET P07949 2/20 0.50
MET P08581 2/20 0.45
SRC P12931 3/20 0.44
CIT O14578 1/20 0.44
GAK O14976 1/20 0.44
EPHB6 O15197 1/20 0.44
ABCC4 O15439 1/20 0.44
DAPK3 O43293 1/20 0.44
RIPK2 O43353 1/20 0.44
NR1I2 O75469 1/20 0.44
RPS6KA4 O75676 1/20 0.44
STK17B O94768 1/20 0.44
STK10 O94804 1/20 0.44
PRKD3 O94806 1/20 0.44
ABCB11 O95342 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31441115 1.00 BRAF (0.64) BRAFRAF1KDREGFRAXL
SCHEMBL21265307 0.87 AXL (0.68) BRAFRAF1KDREGFRAXL
SCHEMBL23749469 0.86 RAF1 (0.62) BRAFRAF1KDREGFRRET
SCHEMBL15084619 0.82 AXL (0.78) BRAFKDREGFRAXLRET
SCHEMBL2744735 0.82 AXL (0.78) BRAFKDREGFRAXLRET
SCHEMBL30001610 0.82 AXL (0.78) BRAFKDREGFRAXLRET
SCHEMBL23749334 0.81 KDR (0.61) BRAFRAF1KDREGFRRET
SCHEMBL23749340 0.81 AXL (0.60) BRAFRAF1KDREGFRAXL
SCHEMBL23749500 0.81 AXL (0.59) BRAFRAF1KDREGFRAXL
SCHEMBL31441112 0.81 AXL (0.59) BRAFRAF1KDREGFRAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3865487-A1 AROMATIC RING-LINKED DIOXANE-QUINAZOLINE OR -QUINOLINE COMPOUNDS, COMPOSITIONS AND USE THEREOF Beijing Scitech-MQ Pharmaceuticals Limited (CN) 2021-08-18 EP disclosed
EP-3865487-A1 AROMATIC RING-LINKED DIOXANE-QUINAZOLINE OR -QUINOLINE COMPOUNDS, COMPOSITIONS AND USE THEREOF Beijing Scitech-MQ Pharmaceuticals Limited (CN) 2021-08-18 EP disclosed