SCHEMBL23763045

SCHEMBL23763045

FC(F)(F)Oc1ccnc(Nc2cc(N3CC4(CCCNC4)C3)nc(-c3cccnc3)n2)c1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 5/20 0.38
ABL1 P00519 2/20 0.38
PIM2 Q9P1W9 1/20 0.38
ROCK2 O75116 2/20 0.36
ROCK1 Q13464 2/20 0.36
CDC42BPA Q5VT25 2/20 0.36
CDC42BPB Q9Y5S2 2/20 0.36
NPY5R Q15761 2/20 0.36
HDAC1 Q13547 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
PIM1 P11309 1/20 0.34
KIT P10721 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29968473 1.00 MAPKAPK2 (0.38) MAPKAPK2ABL1PIM2ROCK2ROCK1
SCHEMBL23763099 0.95 PIM1 (0.38) MAPKAPK2ABL1NPY5RPIM1KIT
SCHEMBL29968465 0.95 PIM1 (0.38) MAPKAPK2ABL1NPY5RPIM1KIT
SCHEMBL29967990 0.95 ALDH1A1 (0.42) MAPKAPK2ABL1PIM2ROCK2ROCK1
SCHEMBL23763037 0.95 ALDH1A1 (0.42) MAPKAPK2ABL1PIM2ROCK2ROCK1
Hydrochloric Acid SCHEMBL29968224 0.95 PIM1 (0.38) MAPKAPK2ABL1NPY5RPIM1KIT
Hydrochloric Acid SCHEMBL29968440 0.94 ALDH1A1 (0.41) MAPKAPK2ABL1PIM2ROCK2ROCK1
SCHEMBL23763087 0.93 PIM1 (0.40) MAPKAPK2ABL1ROCK2ROCK1CDC42BPA
SCHEMBL29968006 0.93 PIM1 (0.40) MAPKAPK2ABL1ROCK2ROCK1CDC42BPA
Hydrochloric Acid SCHEMBL29968459 0.92 PIM1 (0.40) MAPKAPK2ABL1ROCK2ROCK1CDC42BPA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021159993-A1 INHIBITORS OF INTERLEUKIN-1 RECEPTOR ASSOCIATED KINASE (IRAK) /FMS-LIKE RECEPTOR TYROSINE KINASE (FLT3), PHARMACEUTICAL PRODUCTS THEREOF, AND METHODS THEREOF PHARMABLOCK SCIENCES (NANJING) , INC. (CN) 2021-08-19 WO disclosed