SCHEMBL23768855

SCHEMBL23768855

O=C(O)c1cnn(Cc2ccc(N3CC4[C@H](C3)C4(F)F)cn2)c1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BTK Q06187 3/20 0.40
KLKB1 P03952 5/20 0.40
L3MBTL1 Q9Y468 2/20 0.38
HSD17B10 Q99714 1/20 0.35
HPGDS O60760 1/20 0.33
ALKBH2 Q6NS38 1/20 0.33
POLB P06746 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
TAS2R8 Q9NYW2 1/20 0.31
PLA2G4A P47712 1/20 0.31
S1PR1 P21453 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23843089 1.00 BTK (0.40) BTKKLKB1L3MBTL1HSD17B10HPGDS
SCHEMBL23769151 0.86 KLKB1 (0.40) BTKKLKB1
SCHEMBL23769333 0.85 BTK (0.43) BTKKLKB1L3MBTL1HSD17B10HPGDS
SCHEMBL23768871 0.82 CA5A (0.35) KLKB1
SCHEMBL23769219 0.81 L3MBTL1 (0.40) BTKKLKB1L3MBTL1HSD17B10HPGDS
SCHEMBL23754313 0.81 KLKB1 (0.42) BTKKLKB1L3MBTL1HSD17B10POLB
SCHEMBL23843223 0.81 KLKB1 (0.42) BTKKLKB1L3MBTL1HSD17B10POLB
SCHEMBL23754309 0.80 KLKB1 (0.45) BTKKLKB1L3MBTL1HSD17B10POLB
SCHEMBL23754184 0.80 KLKB1 (0.42) BTKKLKB1L3MBTL1HSD17B10HPGDS
SCHEMBL29906534 0.80 KLKB1 (0.42) BTKKLKB1L3MBTL1HSD17B10HPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021160718-A1 HETEROAROMATIC CARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-08-19 WO disclosed