SCHEMBL23769617

SCHEMBL23769617

OCc1cn(Cc2ccc(N3CC4CC4C3)nc2Cl)nn1

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 9/20 0.46
KLKB1 P03952 5/20 0.39
BTK Q06187 4/20 0.38
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
KCNMA1 Q12791 1/20 0.33
DPP4 P27487 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23830178 0.89 KLKB1 (0.39) NOTUMKLKB1BTK
SCHEMBL23769531 0.86 NOTUM (0.43) NOTUMKLKB1KDM4EMAPTKCNMA1
SCHEMBL23769239 0.84 KLKB1 (0.40) NOTUMKLKB1BTKDPP4
SCHEMBL23773107 0.84 KLKB1 (0.44) NOTUMKLKB1BTKDPP4
SCHEMBL23843182 0.82 KLKB1 (0.47) KLKB1BTKDPP4
SCHEMBL23769144 0.80 SMPD3 (0.38) KLKB1
SCHEMBL23769187 0.77 ALDH1A1 (0.52) KLKB1BTK
SCHEMBL23830164 0.76 KLKB1 (0.39) KLKB1BTK
SCHEMBL23830230 0.76 BTK (0.41) KLKB1BTK
SCHEMBL23830171 0.75 KLKB1 (0.39) KLKB1BTKKCNMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021160718-A1 HETEROAROMATIC CARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-08-19 WO disclosed