SCHEMBL23769239

SCHEMBL23769239

CCc1nc(N2CC3CC3C2)ccc1Cn1cc(CO)nn1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 10/20 0.40
NOTUM Q6P988 2/20 0.39
BTK Q06187 5/20 0.37
P2RX7 Q99572 1/20 0.33
DPP4 P27487 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23830164 0.92 KLKB1 (0.39) KLKB1BTK
SCHEMBL23769617 0.84 NOTUM (0.46) KLKB1NOTUMBTKDPP4
SCHEMBL23843156 0.83 KLKB1 (0.47) KLKB1BTK
SCHEMBL23773107 0.82 KLKB1 (0.44) KLKB1NOTUMBTKDPP4
SCHEMBL23830230 0.81 BTK (0.41) KLKB1BTK
SCHEMBL23769616 0.81 SMPD3 (0.36) KLKB1
SCHEMBL23830178 0.80 KLKB1 (0.39) KLKB1NOTUMBTK
SCHEMBL23830171 0.80 KLKB1 (0.39) KLKB1BTK
SCHEMBL23830237 0.78 KLKB1 (0.40) KLKB1BTK
SCHEMBL30087403 0.77 ALDH1A1 (0.48) KLKB1BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021160718-A1 HETEROAROMATIC CARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-08-19 WO disclosed