SCHEMBL23769720

SCHEMBL23769720

CCOC(=O)c1cn(Cc2ccc(N3CCC(C)C3)cc2C#N)cn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 4/20 0.49
NOTUM Q6P988 1/20 0.39
USP30 Q70CQ3 1/20 0.35
MAPT P10636 1/20 0.35
PRKD3 O94806 1/20 0.34
MAP4K4 O95819 1/20 0.34
PIM1 P11309 1/20 0.34
CLK2 P49760 1/20 0.34
MAP4K2 Q12851 1/20 0.34
CAMK2D Q13557 1/20 0.34
DYRK1A Q13627 1/20 0.34
PIM3 Q86V86 1/20 0.34
AURKB Q96GD4 1/20 0.34
PRKD2 Q9BZL6 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
STK17A Q9UEE5 1/20 0.34
MAP4K5 Q9Y4K4 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
P2RY12 Q9H244 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23769721 0.88 NOTUM (0.41) KLKB1NOTUMMAPTPRKD3MAP4K4
SCHEMBL23754054 0.87 KLKB1 (0.60) KLKB1NOTUMP2RY12
SCHEMBL23754350 0.84 KLKB1 (0.62) KLKB1NOTUMMAPT
SCHEMBL29906552 0.84 KLKB1 (0.62) KLKB1NOTUMMAPT
SCHEMBL28986729 0.78 NOTUM (0.53) NOTUMUSP30
SCHEMBL29906606 0.74 KLKB1 (0.46) KLKB1NOTUMMAPTKDM4EALDH1A1
SCHEMBL23754033 0.74 KLKB1 (0.46) KLKB1NOTUMMAPTKDM4EALDH1A1
SCHEMBL29906588 0.73 KLKB1 (0.63) KLKB1
SCHEMBL23754316 0.73 KLKB1 (0.63) KLKB1
SCHEMBL23753990 0.73 KLKB1 (0.45) KLKB1NOTUMMAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021160718-A1 HETEROAROMATIC CARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-08-19 WO disclosed