SCHEMBL23770327

SCHEMBL23770327

CCCOCCNC(=O)COc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O

nearest known ligand 0.69

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 8/20 0.69
DDB1 Q16531 6/20 0.69
HDAC1 Q13547 6/20 0.64
HDAC6 Q9UBN7 6/20 0.64
HDAC3 O15379 2/20 0.64
HDAC2 Q92769 2/20 0.64
MAPT P10636 1/20 0.63
SNCA P37840 1/20 0.63
STAT3 P40763 1/20 0.62
HDAC4 P56524 1/20 0.60
NCOR2 Q9Y618 1/20 0.60
PIP4K2C Q8TBX8 3/20 0.57
TRIM24 O15164 3/20 0.57
BRD4 O60885 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20148960 0.99 CRBN (0.68) CRBNDDB1HDAC1HDAC6HDAC3
SCHEMBL22507973 0.99 CRBN (0.68) CRBNDDB1HDAC1HDAC6HDAC3
SCHEMBL22507989 0.99 CRBN (0.68) CRBNDDB1HDAC1HDAC6HDAC3
SCHEMBL19764205 0.99 CRBN (0.68) CRBNDDB1HDAC1HDAC6HDAC3
SCHEMBL26317544 0.96 CRBN (0.73) CRBNDDB1HDAC1HDAC6HDAC3
SCHEMBL18494154 0.95 CRBN (0.67) CRBNDDB1HDAC1HDAC6HDAC3
SCHEMBL20791883 0.95 CRBN (0.69) CRBNDDB1HDAC1HDAC6HDAC3
SCHEMBL20791890 0.95 CRBN (0.69) CRBNDDB1HDAC1HDAC6HDAC3
SCHEMBL20791887 0.95 CRBN (0.69) CRBNDDB1HDAC1HDAC6HDAC3
SCHEMBL23770363 0.95 CRBN (0.71) CRBNDDB1HDAC1HDAC6HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11708353-B2 Inhibitors of prolyl-tRNA-synthetase THE GENERAL HOSPITAL CORPORATION (US) 2023-07-25 US disclosed
US-20210253558-A1 Inhibitors of Prolyl-tRNA-Synthetase PRESIDENT AND FELLOWS OF HARVARD COLLEGE 2021-08-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11708353-B2 Inhibitors of prolyl-tRNA-synthetase GARS1, AARS1, NSUN3 CRBN 3880/4885DDB1 1306/4885HDAC1 830/4885
US-20210253558-A1 Inhibitors of Prolyl-tRNA-Synthetase GARS1, AARS1, TRMT1 CRBN 3709/4885DDB1 1321/4885HDAC1 805/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.