SCHEMBL23778293

SCHEMBL23778293

CCN(C(=O)O)[C@H]1CCN([C@H]2CC[C@@](C#N)(c3ccc(Cl)cn3)CC2)C1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 2/20 0.39
MCHR1 Q99705 6/20 0.38
CYP2D6 P10635 3/20 0.38
CCR5 P51681 3/20 0.35
HRH3 Q9Y5N1 2/20 0.35
KCNH2 Q12809 1/20 0.35
TACR3 P29371 3/20 0.34
DPP4 P27487 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23778250 1.00 USP30 (0.39) USP30MCHR1CYP2D6CCR5HRH3
SCHEMBL23778248 0.89 CYP2D6 (0.43) USP30MCHR1CYP2D6CCR5HRH3
SCHEMBL23778319 0.85 HSD11B1 (0.45) USP30CYP2D6CCR5HRH3KCNH2
SCHEMBL23778339 0.85 HSD11B1 (0.45) USP30CYP2D6CCR5HRH3KCNH2
SCHEMBL28954172 0.84 CYP2D6 (0.37) USP30MCHR1CYP2D6TACR3
SCHEMBL20066000 0.83 USP30 (0.43) USP30MCHR1CYP2D6HRH3TACR3
SCHEMBL23778331 0.82 CCR5 (0.37) USP30CYP2D6CCR5HRH3KCNH2
SCHEMBL23778432 0.82 CCR5 (0.37) USP30CYP2D6CCR5HRH3KCNH2
SCHEMBL23778286 0.81 CCR5 (0.41) USP30MCHR1CYP2D6CCR5HRH3
SCHEMBL23778237 0.81 CYP2D6 (0.44) USP30MCHR1CYP2D6CCR5HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3526207-B1 HETEROCYCLIC COMPOUNDS HAVING ACTIVITY AS MODULATORS OF MUSCARINIC M1 AND/OR M4 RECEPTORS IN THE TREATMENT OF CNS DISEASES AND PAINS. HEPTARES THERAPEUTICS LTD (GB) 2021-09-08 EP claimed