SCHEMBL23778304

SCHEMBL23778304

Cc1ccc2c(c1)C1(CCC(N3CC[C@H](NC(=O)O)C3)CC1)C(=O)N2

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 6/20 0.43
CCR2 P41597 1/20 0.38
KCNH2 Q12809 1/20 0.38
IP6K1 Q92551 7/20 0.37
IP6K3 Q96PC2 1/20 0.37
IP6K2 Q9UHH9 1/20 0.37
CYP1A2 P05177 2/20 0.36
CYP2C19 P33261 2/20 0.36
POLB P06746 1/20 0.36
CYP3A4 P08684 1/20 0.36
BRD4 O60885 1/20 0.36
RAF1 P04049 1/20 0.36
CYP2C9 P11712 1/20 0.36
CHRM1 P11229 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20073880 0.89 MAPK14 (0.40) MAPK14CCR2KCNH2IP6K1BRD4
SCHEMBL24609136 0.89 MAPK14 (0.40) MAPK14CCR2KCNH2IP6K1BRD4
SCHEMBL23778447 0.88 NQO2 (0.41) MAPK14IP6K1
SCHEMBL21082744 0.83 CCR2 (0.40) MAPK14CCR2KCNH2IP6K1
SCHEMBL23778313 0.82 MAPK14 (0.46) MAPK14CYP1A2CYP2C19RAF1CYP2C9
SCHEMBL20073881 0.82 MAPK14 (0.46) MAPK14CCR2KCNH2CYP1A2CYP2C19
SCHEMBL29709316 0.82 MAPK14 (0.46) MAPK14CCR2KCNH2CYP1A2CYP2C19
SCHEMBL23798012 0.81 MAPK14 (0.45) MAPK14CYP1A2CYP2C19RAF1CYP2C9
SCHEMBL23778317 0.80 MAPK14 (0.40) MAPK14CCR2KCNH2CHRM1
SCHEMBL23778227 0.80 CCR5 (0.38) MAPK14KCNH2IP6K1IP6K3IP6K2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3526207-B1 HETEROCYCLIC COMPOUNDS HAVING ACTIVITY AS MODULATORS OF MUSCARINIC M1 AND/OR M4 RECEPTORS IN THE TREATMENT OF CNS DISEASES AND PAINS. HEPTARES THERAPEUTICS LTD (GB) 2021-09-08 EP disclosed