SCHEMBL23797282

SCHEMBL23797282

C[Si](C)(C)CCOCn1c(-c2ccc(F)cc2)nc(Cl)c1Br

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 4/20 0.40
KDM4E B2RXH2 3/20 0.34
TSHR P16473 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
MAPT P10636 2/20 0.34
THRB P10828 2/20 0.34
TNKS2 Q9H2K2 2/20 0.34
ALDH1A1 P00352 4/20 0.33
HTT P42858 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 1/20 0.32
APOBEC3G Q9HC16 1/20 0.32
F11 P03951 1/20 0.32
CES2 O00748 1/20 0.32
CASR P41180 2/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL68112 0.87 DGAT1 (0.41) DGAT1KDM4ETSHRMEN1KMT2A
SCHEMBL22234417 0.85 DGAT1 (0.40) DGAT1KDM4ETSHRMEN1KMT2A
SCHEMBL23781145 0.82 DGAT1 (0.38) DGAT1KDM4EMEN1KMT2AALDH1A1
SCHEMBL22470948 0.78 MAPK14 (0.44) DGAT1
SCHEMBL23797464 0.77 DGAT1 (0.44) DGAT1KDM4ETSHRMEN1KMT2A
SCHEMBL67447 0.75 DGAT1 (0.40) DGAT1KDM4ETSHRMAPTALDH1A1
SCHEMBL67109 0.75 TNIK (0.43) DGAT1MAPT
SCHEMBL6982067 0.74 DGAT1 (0.58) DGAT1ALDH1A1HPGD
SCHEMBL66909 0.74 DGAT1 (0.47) DGAT1KDM4ETHRBALDH1A1CASR
SCHEMBL68153 0.72 MAPK14 (0.39) DGAT1KDM4EMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3876928-A2 INHIBITORS OF HISTONE DEACETYLASE USEFUL FOR THE TREATMENT OR PREVENTION OF HIV INFECTION Merck Sharp & Dohme Corp. (US) 2021-09-15 EP disclosed