SCHEMBL23797464

SCHEMBL23797464

C[Si](C)(C)CCOCn1c(Br)cnc1-c1ccc(F)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 4/20 0.44
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
KDM4E B2RXH2 2/20 0.35
TSHR P16473 2/20 0.35
MAPT P10636 2/20 0.35
ALDH1A1 P00352 2/20 0.34
HPGD P15428 2/20 0.34
CACNA2D1 P54289 1/20 0.34
PPARD Q03181 2/20 0.34
HSD17B10 Q99714 1/20 0.33
APOBEC3G Q9HC16 1/20 0.33
ELANE P08246 3/20 0.33
ALOX5AP P20292 2/20 0.32
FEN1 P39748 2/20 0.32
NPC1 O15118 1/20 0.31
PTGS2 P35354 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2073673 0.80 DGAT1 (0.41) DGAT1KDM4ETSHRMAPTALDH1A1
SCHEMBL68112 0.79 DGAT1 (0.41) DGAT1MEN1KMT2AKDM4ETSHR
SCHEMBL16828763 0.79 DGAT1 (0.41) DGAT1KMT2AMAPTNPC1
SCHEMBL15572246 0.77 DGAT1 (0.40) DGAT1MAPTNPC1
SCHEMBL22234417 0.77 DGAT1 (0.40) DGAT1MEN1KMT2AKDM4ETSHR
SCHEMBL23797282 0.77 DGAT1 (0.40) DGAT1MEN1KMT2AKDM4ETSHR
SCHEMBL16787698 0.76 DGAT1 (0.50) DGAT1KDM4EMAPTPPARDALOX5AP
SCHEMBL21838857 0.75 DGAT1 (0.41) DGAT1KDM4ETSHRMAPTNPC1
SCHEMBL15986164 0.75 MAPT (0.38) DGAT1KDM4ETSHRMAPTALDH1A1
SCHEMBL31457411 0.75 DGAT1 (0.38) DGAT1MAPTALDH1A1ALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3876928-A2 INHIBITORS OF HISTONE DEACETYLASE USEFUL FOR THE TREATMENT OR PREVENTION OF HIV INFECTION Merck Sharp & Dohme Corp. (US) 2021-09-15 EP disclosed