SCHEMBL23797447

SCHEMBL23797447

BrC=Cc1cc(Br)ccc1Br

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.39
TLR9 Q9NR96 1/20 0.39
ERN1 O75460 1/20 0.39
CA12 O43570 1/20 0.36
CA9 Q16790 1/20 0.36
CYP2A6 P11509 2/20 0.36
ALOX15 P16050 1/20 0.36
S100A4 P26447 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPK1 P28482 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PTPRC P08575 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD11B1 P28845 1/20 0.33
AHR P35869 3/20 0.32
BACE1 P56817 1/20 0.32
AR P10275 1/20 0.32
CASP1 P29466 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23797445 1.00 HSP90AA1 (0.39) HSP90AA1TLR9ERN1CA12CA9
SCHEMBL28702504 0.81 ALOX15 (0.41) HSP90AA1TLR9ERN1CA12CA9
SCHEMBL30464061 0.81 ALOX15 (0.41) HSP90AA1TLR9ERN1CA12CA9
SCHEMBL12205351 0.76 ERN1 (0.35) ERN1CA12CA9CYP2A6ALDH1A1
SCHEMBL16959640 0.73 ERN1 (0.45) HSP90AA1TLR9ERN1CA12CA9
SCHEMBL2787330 0.73 HSP90AA1 (0.41) HSP90AA1TLR9ERN1CA12CA9
SCHEMBL414267 0.73 ERN1 (0.61) HSP90AA1TLR9ERN1CA12CA9
SCHEMBL29661857 0.73 HSP90AA1 (0.41) HSP90AA1TLR9ERN1CA12CA9
SCHEMBL5539045 0.73 ERN1 (0.41) HSP90AA1TLR9ERN1CA12CA9
SCHEMBL5862650 0.73 EIF2AK2 (0.55) HSP90AA1ERN1CA12CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3876928-A2 INHIBITORS OF HISTONE DEACETYLASE USEFUL FOR THE TREATMENT OR PREVENTION OF HIV INFECTION Merck Sharp & Dohme Corp. (US) 2021-09-15 EP disclosed