SCHEMBL23799149

SCHEMBL23799149

COc1ccc2c(c1)NC(=O)C21CCC(N2CCCN(C)CC2)CC1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.41
MAOB P27338 2/20 0.41
PDE7A Q13946 1/20 0.41
OTUD7B Q6GQQ9 1/20 0.41
NPC1 O15118 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MAPK14 Q16539 2/20 0.40
OPRM1 P35372 2/20 0.40
OPRK1 P41145 1/20 0.40
OPRL1 P41146 1/20 0.40
AKR1B1 P15121 1/20 0.39
SIGMAR1 Q99720 2/20 0.39
GHSR Q92847 2/20 0.38
HRH3 Q9Y5N1 1/20 0.38
ACVR1 Q04771 1/20 0.37
FLT3 P36888 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23799162 0.92 FLT3 (0.42) MAOAMAOBPDE7AOTUD7BNPC1
SCHEMBL23778351 0.86 HRH3 (0.42) PDE7AMAPK14HRH3
SCHEMBL20066054 0.83 ALDH1A1 (0.47) MAPK14HRH3
SCHEMBL30179251 0.83 ALDH1A1 (0.47) MAPK14HRH3
SCHEMBL23798701 0.82 OPRM1 (0.51) OPRM1OPRK1OPRL1
SCHEMBL23799175 0.81 PDE7A (0.47) MAOAMAOBPDE7AOTUD7BNPC1
SCHEMBL23798666 0.80 CYP1A2 (0.39) MAPK14OPRM1OPRK1OPRL1AKR1B1
SCHEMBL23798608 0.80 ACVR1 (0.35) MAOAMAOBOTUD7BMAPK14ACVR1
SCHEMBL23798691 0.79 OPRM1 (0.38) MAOAMAOBMAPK14OPRM1OPRK1
SCHEMBL23778269 0.78 HRH3 (0.42) PDE7AHRH3FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3526207-B1 HETEROCYCLIC COMPOUNDS HAVING ACTIVITY AS MODULATORS OF MUSCARINIC M1 AND/OR M4 RECEPTORS IN THE TREATMENT OF CNS DISEASES AND PAINS. HEPTARES THERAPEUTICS LTD (GB) 2021-09-08 EP disclosed