SCHEMBL2381616

SCHEMBL2381616

CCCCC1C(=O)N(c2cccc(C)c2C)CCN1C(Cc1ccc(C#N)cc1)c1cnc[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FNTA P49354 11/20 0.47
FNTB P49356 11/20 0.47
PGGT1B P53609 4/20 0.46
CYP19A1 P11511 2/20 0.34
KCNH2 Q12809 3/20 0.33
ADRA2A P08913 4/20 0.32
ADRA2B P18089 4/20 0.32
ADRA2C P18825 4/20 0.32
ADRA1A P35348 3/20 0.32
ADRA1B P35368 3/20 0.32
ADRA1D P25100 2/20 0.32
TP53 P04637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32
SLC6A2 P23975 1/20 0.32
HTR7 P34969 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL8162228 0.94 FNTA (0.43) FNTAFNTBPGGT1BCYP19A1KCNH2
SCHEMBL4405093 0.94 FNTA (0.40) FNTAFNTBPGGT1BCYP19A1KCNH2
SCHEMBL5551508 0.89 FNTA (0.44) FNTAFNTBPGGT1BKCNH2GRM2
SCHEMBL445626 0.85 FNTA (0.59) FNTAFNTBPGGT1BCYP19A1KCNH2
SCHEMBL3687066 0.85 FNTA (0.59) FNTAFNTBPGGT1BCYP19A1KCNH2
SCHEMBL3517007 0.84 FNTA (0.50) FNTAFNTBPGGT1BCYP19A1KCNH2
Hydrochloric Acid SCHEMBL7818562 0.82 FNTA (0.54) FNTAFNTBPGGT1BCYP19A1KCNH2
Hydrochloric Acid SCHEMBL7837910 0.82 FNTA (0.58) FNTAFNTBPGGT1BCYP19A1KCNH2
SCHEMBL7453424 0.81 FNTA (0.53) FNTAFNTBPGGT1BCYP19A1KCNH2
SCHEMBL7749673 0.81 FNTA (0.53) FNTAFNTBPGGT1BCYP19A1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2547661-A2 INDAZOLE COMPOUNDS AND THEIR USES Dana-Farber Cancer Institute, Inc. (US) 2013-01-23 EP disclosed
WO-2011115725-A2 INDAZOLE COMPOUNDS AND THEIR USES DANA-FARBER CANCER INSTITUTE, INC. (US) 2011-09-22 WO disclosed