SCHEMBL23824151

SCHEMBL23824151

COC(=O)c1n[nH]cc1C(N)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.44
STAT3 P40763 1/20 0.44
HIF1A Q16665 1/20 0.44
NPSR1 Q6W5P4 1/20 0.43
KDM4C Q9H3R0 1/20 0.41
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
MAPK1 P28482 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.36
ALDH1A1 P00352 4/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HSD17B10 Q99714 2/20 0.35
CFTR P13569 1/20 0.35
NNMT P40261 2/20 0.35
GLA P06280 1/20 0.35
GAA P10253 1/20 0.35
MAP2K1 Q02750 1/20 0.35
NR4A2 P43354 1/20 0.34
CREBBP Q92793 1/20 0.34
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL69295 0.86 NPSR1 (0.48) KDM4ESTAT3HIF1ANPSR1KDM4C
SCHEMBL23824150 0.83 NPSR1 (0.45) KDM4ESTAT3HIF1ANPSR1KDM4C
SCHEMBL9799881 0.82 ALDH1A1 (0.34) KDM4ETSHRMAPK1ALDH1A1HSD17B10
SCHEMBL546639 0.77 NPSR1 (0.46) KDM4ESTAT3HIF1ANPSR1KDM4C
SCHEMBL19763311 0.75 KDM4C (0.48) KDM4ESTAT3HIF1ANPSR1KDM4C
SCHEMBL5761874 0.75 NPSR1 (0.48) KDM4ESTAT3HIF1ANPSR1KDM4C
SCHEMBL19207970 0.73 NPSR1 (0.46) KDM4ESTAT3HIF1ANPSR1KDM4C
SCHEMBL20168105 0.73 NNMT (0.41) KDM4EALDH1A1NNMTGLAGAA
SCHEMBL19780563 0.73 NPSR1 (0.46) KDM4ESTAT3HIF1ANPSR1KDM4C
SCHEMBL13726965 0.73 NPSR1 (0.46) KDM4ESTAT3HIF1ANPSR1KDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021181122-A1 GPR52 MODULATOR COMPOUNDS HEPTARES THERAPEUTICS LIMITED (GB) 2021-09-16 WO disclosed